SCHEMBL3475398

SCHEMBL3475398

CC(C)(C)Cn1nnc2c(Br)c(-c3cncc(C#N)c3)ccc21

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 3/20 0.33
USP7 Q93009 2/20 0.33
P4HTM Q9NXG6 1/20 0.33
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
CDC42BPB Q9Y5S2 1/20 0.32
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
CYP1A2 P05177 1/20 0.32
METAP2 P50579 1/20 0.32
AR P10275 1/20 0.31
BACE1 P56817 1/20 0.31
KCNH2 Q12809 1/20 0.31
GRIN1 Q05586 2/20 0.31
GRIN2B Q13224 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3475357 0.86 GRM2 (0.43) GRM2
SCHEMBL3476240 0.85 GRM2 (0.39) GRM2CYP11B2
SCHEMBL3475355 0.84 GRM2 (0.35) GRM2CYP11B1CYP11B2GRIN1GRIN2B
SCHEMBL3476991 0.82 GRM2 (0.35) GRM2
SCHEMBL7808336 0.82 CYP11B1 (0.39) GRM2CYP11B1CYP11B2CYP1A2
SCHEMBL3476696 0.80 GRM2 (0.37) GRM2ARGRIN2B
SCHEMBL3469755 0.79 CNR1 (0.37) GRM2P4HTMCYP11B1CYP1A2
SCHEMBL3475412 0.79 GRM2 (0.33) GRM2AR
SCHEMBL3475817 0.78 GRM2 (0.36) GRM2
SCHEMBL3474766 0.77 GRM2 (0.39) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO claimed
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO disclosed
WO-2010141360-A1 BIARYL BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2010-12-09 WO disclosed