SCHEMBL7808601

SCHEMBL7808601

Nc1ncc(CN2CCN(c3cccc(Cl)c3)CC2)c(N)n1

nearest known ligand 0.72

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DHFR P00374 8/20 0.72
DRD4 P21917 2/20 0.55
DRD3 P35462 1/20 0.55
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
MAPT P10636 1/20 0.51
GAA P10253 1/20 0.50
GFER P55789 1/20 0.50
KCNH2 Q12809 1/20 0.50
KDM4E B2RXH2 1/20 0.49
OPRM1 P35372 1/20 0.49
OPRD1 P41143 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7802247 0.88 DHFR (0.57) DHFRDRD4DRD3ALDH1A1LMNA
Hydrochloric Acid SCHEMBL7806908 0.87 DHFR (0.56) DHFRDRD4DRD3ALDH1A1LMNA
SCHEMBL7810190 0.85 DHFR (0.65) DHFRDRD4DRD3ALDH1A1LMNA
SCHEMBL7807168 0.85 DHFR (0.70) DHFRDRD4DRD3ALDH1A1LMNA
Hydrochloric Acid SCHEMBL7813876 0.84 DHFR (0.64) DHFRDRD4DRD3ALDH1A1LMNA
Hydrochloric Acid SCHEMBL7811194 0.84 DHFR (0.69) DHFRDRD4DRD3ALDH1A1LMNA
SCHEMBL7801857 0.80 ALDH1A1 (0.61) DHFRDRD4DRD3ALDH1A1MAPT
SCHEMBL7807221 0.78 DHFR (0.65) DHFRDRD4DRD3LMNA
Hydrochloric Acid SCHEMBL7807039 0.77 DHFR (0.64) DHFRALDH1A1MAPT
SCHEMBL7810326 0.76 DHFR (0.59) DHFRDRD4ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0873317-B1 PYRIMIDIN DERIVATIVES HOFFMANN LA ROCHE (CH) 2001-04-11 EP disclosed
EP-0873317-A1 PYRIMIDIN DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1998-10-28 EP disclosed
US-5688798-A PSYCHOTIC ILLNESS SUCH AS SCHIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1997-11-18 US disclosed
WO-1997013759-A1 PYRIMIDIN DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-04-17 WO disclosed