SCHEMBL7808799

SCHEMBL7808799

CS(=O)(=O)c1ccc(/C(=C2\CCOC2=O)c2ccc(F)c(Cl)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.46
PTGS1 P23219 6/20 0.46
PROKR1 Q8TCW9 1/20 0.37
AKR1C3 P42330 1/20 0.37
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7808801 1.00 PTGS2 (0.46) PTGS2PTGS1PROKR1AKR1C3ADORA3
SCHEMBL7811301 0.90 PTGS2 (0.43) PTGS2PTGS1AKR1C3ADORA3ADORA2A
SCHEMBL7807030 0.90 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL7802244 0.90 PTGS2 (0.43) PTGS2PTGS1AKR1C3ADORA3ADORA2A
SCHEMBL7807028 0.90 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL7806923 0.90 PTGS2 (0.43) PTGS2PTGS1AKR1C3ADORA3ADORA2A
SCHEMBL7802217 0.89 PTGS1 (0.46) PTGS2PTGS1
SCHEMBL7802214 0.89 PTGS1 (0.46) PTGS2PTGS1
SCHEMBL1782770 0.87 PTGS2 (0.46) PTGS2PTGS1AKR1C3ADORA3ADORA2A
SCHEMBL7806930 0.87 PTGS2 (0.46) PTGS2PTGS1AKR1C3ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891345-B1 NOVEL FURAN DIARYLMETHYLIDENE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THERAPEUTICAL USES THEREOF UNION PHARMA SCIENT APPL (FR) 2001-08-16 EP disclosed
US-6180651-B1 ANTIINFLAMMATORY AGENTS; ANALGESICS BRISTOL-MYERS SQUIBB 2001-01-30 US disclosed
WO-2000014082-A1 DIARYLMETHYLIDENE FURAN DERIVATIVES AS DRUGS WITH ANTI-INFLAMMATORY, ANALGESIC AND CHEMOPREVENTIVE PROPERTIES LABORATORIES UPSA (FR) 2000-03-16 WO disclosed