SCHEMBL7809537

SCHEMBL7809537

CN1C(=O)C(NC(=O)Nc2cccc(I)c2)N=C(N2CC3CCC(CC3)C2)c2ccccc21

nearest known ligand 0.82

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 20/20 0.82
CCKAR P32238 2/20 0.68
KCNH2 Q12809 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7817088 1.00 CCKBR (0.82) CCKBRCCKARKCNH2
SCHEMBL7824899 0.91 CCKBR (0.84) CCKBR
L-740093 SCHEMBL31616330 0.90 CCKBR (1.00) CCKBRKCNH2
L-740093 SCHEMBL5198570 0.90 CCKBR (1.00) CCKBRKCNH2
L-740093 SCHEMBL7627122 0.90 CCKBR (1.00) CCKBRKCNH2
L-740093 SCHEMBL7818686 0.90 CCKBR (1.00) CCKBRKCNH2
SCHEMBL7816266 0.90 CCKBR (0.82) CCKBRKCNH2
SCHEMBL7817950 0.90 CCKBR (0.82) CCKBRKCNH2
Hydrochloric Acid SCHEMBL7819113 0.89 CCKBR (0.82) CCKBRKCNH2
SCHEMBL7816438 0.87 CCKBR (0.79) CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0652871-B1 BENZODIAZEPINE DERIVATIVES MERCK SHARP & DOHME (GB) 2001-10-17 EP claimed
US-5618812-A GASTRIN ANTAGONISTS; GASTROINTESTINAL DISORDERS MERCK SHARP & DOHME, LTD. (GB) 1997-04-08 US claimed
WO-1994003437-A1 BENZODIAZEPINE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1994-02-17 WO claimed
EP-0652871-B1 BENZODIAZEPINE DERIVATIVES MERCK SHARP & DOHME (GB) 2001-10-17 EP disclosed
US-5618812-A GASTRIN ANTAGONISTS; GASTROINTESTINAL DISORDERS MERCK SHARP & DOHME, LTD. (GB) 1997-04-08 US disclosed
WO-1994003437-A1 BENZODIAZEPINE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1994-02-17 WO disclosed