SCHEMBL7809974

SCHEMBL7809974

C[SiH](C)O[C@@H](CC(C)(C)C)c1ccccc1Br

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
CYP2C19 P33261 2/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32
HTT P42858 1/20 0.32
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4610096 0.75 IDO1 (0.35) IDO1TDO2CYP2C19ALDH1A1CYP3A4
SCHEMBL7765110 0.73 GAA (0.32)
SCHEMBL6160182 0.72 SLC6A2 (0.37) IDO1TDO2ALDH1A1CYP3A4
SCHEMBL1093213 0.68 RIPK1 (0.38) IDO1TDO2CYP2C19ALDH1A1CYP3A4
SCHEMBL9701751 0.68
SCHEMBL13465755 0.66 CYP2C19 (0.43) CYP2C19ALDH1A1CYP3A4ALOX15HTT
SCHEMBL8069568 0.66 RIPK1 (0.37) ALDH1A1
SCHEMBL5872179 0.66 MEN1 (0.37)
SCHEMBL8879657 0.64 TYR (0.42) ALDH1A1
SCHEMBL5847735 0.63 CYP2C19 (0.42) IDO1TDO2CYP2C19ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1075467-A1 PYRAZOLE DERIVATIVES AS P-38 MAP KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2001-02-14 EP disclosed
WO-1999057101-A1 PYRAZOLE DERIVATIVES AS P-38 MAP KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 1999-11-11 WO disclosed