SCHEMBL7810052

SCHEMBL7810052

N#Cc1cccc(-c2nc(-c3ccc4ccccc4c3)c[nH]2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.46
XDH P47989 1/20 0.44
ALDH1A3 P47895 1/20 0.42
PGR P06401 1/20 0.42
CYP17A1 P05093 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
PIN1 Q13526 1/20 0.41
TYMP P19971 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
GABRG2 P18507 2/20 0.41
GABRB3 P28472 2/20 0.41
GABRA5 P31644 2/20 0.41
GABRA3 P34903 2/20 0.41
GABRA1 P14867 1/20 0.41
PIM1 P11309 1/20 0.41
MAOB P27338 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
ADORA2A P29274 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27544569 0.89 GABRG2 (0.51) IDO1XDHALDH1A3PIN1TYMP
SCHEMBL7141999 0.87 IDO1 (0.51) IDO1XDHALDH1A3PIN1CLK4
SCHEMBL7809837 0.83 PTGDR (0.48) IDO1CYP11B1CYP11B2PIN1CLK4
SCHEMBL5128314 0.82 CYP1A1 (0.56) CYP17A1CYP11B1CYP11B2ADORA2AADORA1
SCHEMBL31305440 0.82 CYP1A1 (0.56) CYP17A1CYP11B1CYP11B2ADORA2AADORA1
SCHEMBL7143474 0.82 GABRG2 (0.53) IDO1XDHALDH1A3CLK4GABRG2
SCHEMBL2950013 0.81 CYP1A1 (0.53) CYP17A1CYP11B1CYP11B2ADORA2AADORA1
SCHEMBL4855853 0.81 CYP1A1 (0.49) CYP17A1CYP11B1CYP11B2MAOB
SCHEMBL31305475 0.81 CYP1A1 (0.53) CYP17A1CYP11B1CYP11B2ADORA2AADORA1
SCHEMBL8118629 0.80 GABRG2 (0.51) IDO1XDHALDH1A3GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed