SCHEMBL7810093

SCHEMBL7810093

CC(C)(Oc1ccccc1N1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1)C(=O)O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.62
KMT2A Q03164 4/20 0.62
SMN1; SMN2 Q16637 4/20 0.62
LMNA P02545 3/20 0.62
NPSR1 Q6W5P4 3/20 0.62
POLB P06746 2/20 0.62
TSHR P16473 2/20 0.62
NPY2R P49146 1/20 0.52
RBP4 P02753 1/20 0.51
SIGMAR1 Q99720 1/20 0.51
HTT P42858 3/20 0.51
GAA P10253 2/20 0.51
MAPT P10636 2/20 0.51
XBP1 P17861 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
HTR1A P08908 1/20 0.50
ADRA1D P25100 1/20 0.50
ADRA1A P35348 1/20 0.50
ADRA1B P35368 1/20 0.50
TACR3 P29371 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7810154 0.90 MEN1 (0.60) MEN1KMT2ASMN1; SMN2LMNANPSR1
SCHEMBL7813944 0.90 MEN1 (0.61) MEN1KMT2ASMN1; SMN2LMNANPSR1
SCHEMBL7811604 0.88 SMN1; SMN2 (0.66) MEN1KMT2ASMN1; SMN2LMNANPSR1
SCHEMBL7810142 0.88 POLB (0.60) MEN1KMT2ASMN1; SMN2LMNANPSR1
SCHEMBL7810164 0.87 MEN1 (0.58) MEN1KMT2ASMN1; SMN2LMNANPSR1
SCHEMBL7813588 0.87 TSHR (0.58) MEN1KMT2ASMN1; SMN2LMNANPSR1
SCHEMBL7814258 0.87 TSHR (0.61) MEN1KMT2ASMN1; SMN2LMNANPSR1
SCHEMBL7810112 0.86 MEN1 (0.64) MEN1KMT2ASMN1; SMN2LMNANPSR1
SCHEMBL7813768 0.80 MEN1 (0.51) MEN1KMT2ASMN1; SMN2LMNANPSR1
SCHEMBL7817538 0.80 PPARD (0.68) MEN1KMT2ASMN1; SMN2NPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0607536-B1 Arylamide derivatives SS PHARMACEUTICAL CO (JP) 2001-01-24 EP disclosed
US-5532371-A SIDE EFFECT REDUCTION SS PHARMACEUTICAL CO., LTD. (JP) 1996-07-02 US disclosed
US-5411972-A Arylamide derivatives for treating hyperlipemia SS PHARMACEUTICAL CO., LTD. (JP) 1995-05-02 US disclosed
EP-0607536-A1 Arylamide derivatives SS PHARMACEUTICAL CO., LTD. (JP) 1994-07-27 EP disclosed