SCHEMBL7811255

SCHEMBL7811255

CN(C(=O)CC(CCOS(C)(=O)=O)c1ccc(Cl)c(Cl)c1)c1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
ALDH1A1 P00352 1/20 0.35
UTS2R Q9UKP6 2/20 0.34
FFAR1 O14842 1/20 0.34
LMNA P02545 1/20 0.33
TACR2 P21452 1/20 0.33
PRKCZ Q05513 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7802907 0.92 ALDH1A1 (0.44) ALDH1A1FFAR1TACR2SLC6A2SLC6A4
SCHEMBL8799934 0.88 ALDH1A1 (0.41) ALDH1A1TACR2SLC6A2SLC6A4SLC6A3
SCHEMBL7807766 0.86 DRD4 (0.41) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL7803020 0.83 ALDH1A1 (0.39) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL8835963 0.80 FNTA (0.49) LMNASLC6A2
SCHEMBL7807795 0.80 PRKCZ (0.47) ALDH1A1FFAR1LMNAPRKCZ
SCHEMBL9318213 0.78 TACR2 (0.47) TACR2
SCHEMBL7807586 0.78 TACR1 (0.41) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL7815271 0.76 TACR2 (0.48) TACR2
SCHEMBL7815376 0.75 FFAR1 (0.40) ALDH1A1UTS2RFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773929-B1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORP (US) 2001-10-31 EP disclosed
US-5654316-A Piperidine derivatives as neurokinin antagonists SCHERING CORPORATION (US) 1997-08-05 US disclosed