SCHEMBL7812415

SCHEMBL7812415

CN(C)C=C(C#N)S(=O)(=O)c1ccccn1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 5/20 0.56
LMNA P02545 3/20 0.54
ALDH1A1 P00352 5/20 0.53
MAPT P10636 1/20 0.53
KMT2A Q03164 4/20 0.52
POLB P06746 1/20 0.52
MAPK1 P28482 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.38
RAB9A P51151 3/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
MEN1 O00255 2/20 0.36
NPC1 O15118 1/20 0.36
MITF O75030 1/20 0.36
HPGD P15428 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.35
ATM Q13315 1/20 0.35
NFE2L2 Q16236 2/20 0.35
TXNRD1 Q16881 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7135383 0.77 PKM (0.54) PKMLMNAALDH1A1MAPTKMT2A
SCHEMBL7135386 0.77 PKM (0.54) PKMLMNAALDH1A1MAPTKMT2A
SCHEMBL17730555 0.77 PKM (0.54) PKMLMNAALDH1A1MAPTKMT2A
SCHEMBL4699004 0.75 PKM (0.65) PKMLMNAALDH1A1MAPTKMT2A
SCHEMBL4699000 0.75 PKM (0.65) PKMLMNAALDH1A1MAPTKMT2A
SCHEMBL5363714 0.74 PKM (0.60) PKMLMNAALDH1A1MAPTKMT2A
SCHEMBL5363709 0.74 PKM (0.60) PKMLMNAALDH1A1MAPTKMT2A
SCHEMBL5363715 0.74 PKM (0.60) PKMLMNAALDH1A1MAPTKMT2A
SCHEMBL8429766 0.72 LMNA (0.52) PKMLMNAALDH1A1MAPTKMT2A
SCHEMBL8429769 0.72 LMNA (0.52) PKMLMNAALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1119566-A1 NOVEL HETEROCYCLYL-METHYL-SUBSTITUTED PYRAZOLES Bayer Aktiengesellschaft (DE) 2001-08-01 EP disclosed
WO-2000021954-A1 NOVEL HETEROCYCLYL-METHYL-SUBSTITUTED PYRAZOLES BAYER AKTIENGESELLSCHAFT (DE) 2000-04-20 WO disclosed