SCHEMBL7813005

SCHEMBL7813005

O=C(O)c1csc(C(=O)CBr)c1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 0.52
DAO P14920 7/20 0.47
PTPN1 P18031 3/20 0.41
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
ALAD P13716 1/20 0.36
HDAC4 P56524 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11167795 0.83 GSK3B (0.50) GSK3BPTPN1CES2CES1
SCHEMBL71474 0.79 DAO (0.58) GSK3BDAOCES2CES1ALAD
SCHEMBL939177 0.79 GSK3B (0.46) GSK3B
SCHEMBL11161465 0.79 GSK3B (0.46) GSK3BDAOPTPN1CES2CES1
SCHEMBL15282434 0.78 GSK3B (0.68) GSK3BDAOPTPN1CES2CES1
SCHEMBL6198736 0.76 CA12 (0.45) GSK3B
SCHEMBL25184460 0.76 GSK3B (0.50) GSK3BPTPN1CES2CES1
SCHEMBL22953102 0.74 GSK3B (0.48) GSK3BPTPN1CES2CES1ALAD
SCHEMBL15547606 0.74 DAO (0.59) GSK3BDAOCES2CES1
SCHEMBL5350815 0.74 DAO (0.57) GSK3BDAOCES2CES1ALAD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0816352-B1 Bi-aryl heterocyclic compounds and their use in human or veterinary medicine and in cosmetics CT INTERNAT DE (FR) 2001-02-21 EP disclosed
EP-0816352-A1 Bi-aryl heterocyclic compounds and their use in human or veterinary medicine and in cosmetics CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (C.I.R.D. GALDERMA) (FR) 1998-01-07 EP disclosed