SCHEMBL7813702

SCHEMBL7813702

COCc1nc2cc(Oc3ccccc3)ccc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 5/20 0.53
GRIN2B Q13224 5/20 0.53
RAB9A P51151 9/20 0.51
NPC1 O15118 8/20 0.51
SMN1; SMN2 Q16637 7/20 0.51
TP53 P04637 3/20 0.51
TSHR P16473 1/20 0.51
ALDH1A1 P00352 1/20 0.50
XDH P47989 1/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
GAA P10253 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
POLB P06746 1/20 0.44
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7813706 0.89 GRIN1 (0.67) GRIN1GRIN2BRAB9ANPC1SMN1; SMN2
SCHEMBL7807068 0.83 GRIN1 (0.56) GRIN1GRIN2BRAB9ANPC1SMN1; SMN2
SCHEMBL7808653 0.83 GRIN1 (0.56) GRIN1GRIN2BRAB9ANPC1SMN1; SMN2
SCHEMBL7806900 0.83 GRIN1 (0.56) GRIN1GRIN2BRAB9ANPC1SMN1; SMN2
SCHEMBL7808790 0.83 GRIN1 (0.56) GRIN1GRIN2BRAB9ANPC1SMN1; SMN2
SCHEMBL7806889 0.82 GRIN1 (0.52) GRIN1GRIN2BRAB9ANPC1SMN1; SMN2
Hydrochloric Acid SCHEMBL8474413 0.82 GRIN1 (0.55) GRIN1GRIN2BRAB9ANPC1SMN1; SMN2
SCHEMBL7810205 0.81 RAB9A (0.56) GRIN1GRIN2BRAB9ANPC1SMN1; SMN2
Hydrochloric Acid SCHEMBL8479280 0.81 GRIN1 (0.51) GRIN1GRIN2BRAB9ANPC1SMN1; SMN2
SCHEMBL7808614 0.80 GRIN1 (0.52) GRIN1GRIN2BRAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820990-B1 Benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR (FR) 2001-01-17 EP disclosed
US-5972968-A INTERLEUKIN INHIBITOR ADIR ET COMPAGNIE (FR) 1999-10-26 US disclosed
EP-0820990-A2 Novel benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR ET COMPAGNIE (FR) 1998-01-28 EP disclosed