SCHEMBL7814637

SCHEMBL7814637

CC(=O)OCC(CCn1cnc2c(SCc3ccccc3)nc(N)nc21)COC(C)=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.59
CYP2C19 P33261 5/20 0.59
CYP2C9 P11712 4/20 0.59
HIF1A Q16665 4/20 0.59
CYP3A4 P08684 3/20 0.59
ALDH1A1 P00352 2/20 0.59
PHLPP2 Q6ZVD8 1/20 0.59
KDM4E B2RXH2 1/20 0.56
HPGD P15428 1/20 0.56
ADRA1A P35348 1/20 0.56
HSD17B10 Q99714 1/20 0.56
RXFP1 Q9HBX9 1/20 0.56
CYP2D6 P10635 3/20 0.52
SLC29A1 Q99808 7/20 0.49
TP53 P04637 1/20 0.41
HK1 P19367 1/20 0.40
HKDC1 Q2TB90 1/20 0.40
MPO P05164 1/20 0.39
HRH4 Q9H3N8 1/20 0.38
ADORA2A P29274 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7816726 0.92 ALDH1A1 (0.55) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7819883 0.86 ALDH1A1 (0.52) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7806581 0.85 ALDH1A1 (0.56) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7806679 0.84 CYP1A2 (0.60) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL6317462 0.81 ALDH1A1 (0.56) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL14163777 0.80 KDM4E (0.69) CYP2C19ALDH1A1KDM4EHPGDADRA1A
SCHEMBL30114962 0.79 KDM4E (0.67) CYP2C19ALDH1A1KDM4EHPGDADRA1A
SCHEMBL3155583 0.79 KDM4E (0.67) CYP2C19ALDH1A1KDM4EHPGDADRA1A
SCHEMBL7813547 0.78 KDM4E (0.66) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7806600 0.78 CYP1A2 (0.59) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0352953-B1 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 2001-01-03 EP claimed
EP-0352953-B1 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 2001-01-03 EP disclosed
US-5017701-A Process for the preparation of purine derivatives BEECHAM GROUP, P.L.C. (GB) 1991-05-21 US disclosed
EP-0352953-A2 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 1990-01-31 EP disclosed