SCHEMBL7806679

SCHEMBL7806679

CCOC(=O)C(CCn1cnc2c(SCc3ccccc3)nc(N)nc21)C(=O)OCC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.60
CYP2C19 P33261 5/20 0.60
CYP2C9 P11712 4/20 0.60
HIF1A Q16665 4/20 0.60
CYP3A4 P08684 3/20 0.60
ALDH1A1 P00352 2/20 0.60
PHLPP2 Q6ZVD8 1/20 0.60
CYP2D6 P10635 3/20 0.56
SLC29A1 Q99808 7/20 0.52
NPC1 O15118 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
RAB9A P51151 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TP53 P04637 1/20 0.41
HK1 P19367 1/20 0.40
HKDC1 Q2TB90 1/20 0.40
MPO P05164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7814637 0.84 CYP1A2 (0.59) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7806600 0.84 CYP1A2 (0.59) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL13645718 0.79 HSP90AB1 (0.51) CYP2C19
SCHEMBL7816726 0.78 ALDH1A1 (0.55) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL28451668 0.77 HSP90AB1 (0.49) CYP2C19
SCHEMBL17595248 0.76 CYP1A2 (1.00) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL7806517 0.72 CYP1A2 (0.59) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL3156963 0.71 KDM4E (0.67) CYP2C19ALDH1A1
SCHEMBL7819883 0.71 ALDH1A1 (0.52) CYP1A2CYP2C19CYP2C9HIF1ACYP3A4
SCHEMBL10917478 0.70 HSP90AB1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0352953-B1 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 2001-01-03 EP disclosed
US-5017701-A Process for the preparation of purine derivatives BEECHAM GROUP, P.L.C. (GB) 1991-05-21 US disclosed
EP-0352953-A2 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 1990-01-31 EP disclosed