SCHEMBL7815736

SCHEMBL7815736

O=C(O)O[C@@H]1CCCN(CCCN2c3ccccc3-c3ccccc3-c3ccccc32)C1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.56
CHRNB4 P30926 1/20 0.56
CHRNA3 P32297 1/20 0.56
CHRNA4 P43681 1/20 0.56
SLC6A1 P30531 3/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7813228 1.00 CHRNB2 (0.56) CHRNB2CHRNB4CHRNA3CHRNA4SLC6A1
SCHEMBL8202527 0.89 CHRNB2 (0.52) CHRNB2CHRNB4CHRNA3CHRNA4SLC6A1
SCHEMBL8206721 0.88 SLC6A1 (0.61) CHRNB2CHRNB4CHRNA3CHRNA4SLC6A1
SCHEMBL8202612 0.88 SLC6A1 (0.61) CHRNB2CHRNB4CHRNA3CHRNA4SLC6A1
SCHEMBL8202368 0.87 SLC6A1 (0.57) CHRNB2CHRNB4CHRNA3CHRNA4SLC6A1
SCHEMBL8203622 0.87 CHRNB2 (0.47) CHRNB2CHRNB4CHRNA3CHRNA4SLC6A1
SCHEMBL8203132 0.87 SLC6A1 (0.61) SLC6A1CYP2D6
SCHEMBL8206888 0.85 SLC6A1 (0.61) CHRNB2CHRNB4CHRNA3CHRNA4SLC6A1
SCHEMBL8206144 0.85 CHRNB2 (0.46) CHRNB2CHRNB4CHRNA3CHRNA4SLC6A1
SCHEMBL7843283 0.84 SLC6A1 (0.52) CHRNB2CHRNB4CHRNA3CHRNA4SLC6A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869954-B1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF NEUROGENIC INFLAMMATION NOVO NORDISK AS (DK) 2001-09-19 EP claimed