SCHEMBL7816730

SCHEMBL7816730

Nc1nc(-c2nn(Cc3ccccc3F)c3ccccc23)ncc1-c1ccccn1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BUB1 O43683 18/20 0.54
ADORA2A P29274 1/20 0.50
ADORA1 P30542 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14843837 0.83 BUB1 (0.67) BUB1
SCHEMBL14843520 0.80 BUB1 (0.68) BUB1
SCHEMBL6214026 0.79 BUB1 (0.53) BUB1
SCHEMBL18212218 0.78 ADORA3 (0.58)
Etriciguat SCHEMBL29388720 0.77 ADORA3 (0.56) BUB1
Etriciguat SCHEMBL419874 0.77 ADORA3 (0.56) BUB1
SCHEMBL4245462 0.76 BUB1 (0.48) BUB1
SCHEMBL174189 0.76 ADORA3 (0.61)
SCHEMBL16101234 0.75 BUB1 (0.60) BUB1
SCHEMBL16096773 0.75 BUB1 (0.55) BUB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1119566-A1 NOVEL HETEROCYCLYL-METHYL-SUBSTITUTED PYRAZOLES Bayer Aktiengesellschaft (DE) 2001-08-01 EP disclosed
WO-2000021954-A1 NOVEL HETEROCYCLYL-METHYL-SUBSTITUTED PYRAZOLES BAYER AKTIENGESELLSCHAFT (DE) 2000-04-20 WO disclosed