SCHEMBL7818136

SCHEMBL7818136

CCOC(=O)C1CN(C)c2cc(C(F)(F)F)ccc2O1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.57
CYP2C9 P11712 2/20 0.57
CYP2C19 P33261 2/20 0.57
CYP3A4 P08684 1/20 0.57
RECQL P46063 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
POLB P06746 2/20 0.52
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.45
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
SIRT2 Q8IXJ6 2/20 0.42
SIRT1 Q96EB6 2/20 0.42
HPGD P15428 1/20 0.41
KDM4E B2RXH2 1/20 0.41
HSP90AA1 P07900 1/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
RORC P51449 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7810147 0.84 POLB (0.55) ALDH1A1CYP2C9CYP2C19CYP3A4RECQL
SCHEMBL7818619 0.84 ALDH1A1 (0.58) ALDH1A1CYP2C9CYP2C19CYP3A4RECQL
SCHEMBL537789 0.83 POLB (0.53) ALDH1A1CYP2C9CYP2C19CYP3A4RECQL
SCHEMBL7818287 0.82 POLB (0.73) ALDH1A1CYP2C9CYP2C19CYP3A4RECQL
SCHEMBL7820037 0.81 POLB (0.53) ALDH1A1NPSR1POLBKMT2AMEN1
SCHEMBL7810528 0.81 POLB (0.54) ALDH1A1CYP2C9CYP2C19CYP3A4RECQL
SCHEMBL7817587 0.81 POLB (0.54) ALDH1A1CYP2C9CYP2C19CYP3A4RECQL
SCHEMBL7808798 0.81 ALDH1A1 (0.60) ALDH1A1CYP2C9CYP2C19CYP3A4RECQL
SCHEMBL17447947 0.81 POLB (0.50) ALDH1A1CYP2C9CYP2C19CYP3A4RECQL
SCHEMBL31343599 0.79 SIRT2 (0.49) ALDH1A1CYP2C9CYP2C19CYP3A4RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894796-B1 Imidazolines substituted with a heterocyclic ring as alpha-2 antagonists ADIR (FR) 2001-06-06 EP disclosed
US-6057317-A Heterocyclic compounds ADIR ET COMPAGNIE (FR) 2000-05-02 US disclosed
EP-0894796-A1 Imidazolines substituted with a heterocyclic ring as alpha-2 antagonists ADIR ET COMPAGNIE (FR) 1999-02-03 EP disclosed