SCHEMBL7818288

SCHEMBL7818288

CC[Si](CC)(CC)O[C@H]1C(=O)N(C(=O)OC(C)(C)C)C1c1ccco1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 11/20 0.40
LMNA P02545 1/20 0.38
KDM4E B2RXH2 2/20 0.36
POLB P06746 1/20 0.36
APEX1 P27695 1/20 0.36
ESR2 Q92731 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 1/20 0.36
RECQL P46063 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LIPE Q05469 1/20 0.35
NR1I2 O75469 1/20 0.35
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ADORA2A P29274 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6394870 1.00 ADORA2B (0.40) ADORA2BLMNAKDM4EPOLBAPEX1
SCHEMBL6394866 1.00 ADORA2B (0.40) ADORA2BLMNAKDM4EPOLBAPEX1
SCHEMBL6839247 1.00 ADORA2B (0.40) ADORA2BLMNAKDM4EPOLBAPEX1
SCHEMBL6861590 0.88 ADORA2B (0.48) ADORA2BLMNAKDM4EPOLBAPEX1
SCHEMBL6861588 0.88 ADORA2B (0.48) ADORA2BLMNAKDM4EPOLBAPEX1
SCHEMBL6861594 0.88 ADORA2B (0.48) ADORA2BLMNAKDM4EPOLBAPEX1
SCHEMBL6858809 0.87 ADORA2B (0.40) ADORA2BLMNAKDM4EPOLBAPEX1
SCHEMBL6858812 0.87 ADORA2B (0.40) ADORA2BLMNAKDM4EPOLBAPEX1
SCHEMBL6858807 0.87 ADORA2B (0.40) ADORA2BLMNAKDM4EPOLBAPEX1
SCHEMBL4334217 0.85 LIPE (0.35) ADORA2BPOLBL3MBTL1LIPENR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0694539-B1 7-O-Ethers of taxane derivatives BRISTOL MYERS SQUIBB CO (US) 2001-11-28 EP disclosed
US-6201140-B1 ANTITUMOR AGENTS BRISTOL-MYERS SQUIBB COMPANY 2001-03-13 US disclosed
EP-0694539-A1 7-o-Ethers of taxane derivatives BRISTOL-MYERS SQUIBB COMPANY (US) 1996-01-31 EP disclosed