SCHEMBL78190

SCHEMBL78190

CC(=O)C1CN(C(=O)OCc2ccccc2)C(CO[Si](C)(C)C(C)(C)C)CC1=O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
PARP1 P09874 1/20 0.38
AGTR2 P50052 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78783 0.86 PDK1 (0.39) PDK1PDK2PDK3PDK4PSEN1
SCHEMBL8701756 0.83 PSEN1 (0.41) PDK1PDK2PDK3PDK4PSEN1
SCHEMBL8701755 0.83 PSEN1 (0.41) PDK1PDK2PDK3PDK4PSEN1
SCHEMBL30781570 0.82 POLB (0.44) PDK1PDK2PDK3PDK4AGTR2
SCHEMBL29560191 0.81 SMN1; SMN2 (0.45) PDK1PDK2PDK3PDK4
SCHEMBL78361 0.81 PARP1 (0.43) PDK1PDK2PDK3PDK4PARP1
SCHEMBL1058639 0.81 POLB (0.49) PDK1PDK2PDK3PDK4PSEN1
SCHEMBL15341340 0.81 PDK1 (0.45) PDK1PDK2PDK3PDK4AGTR2
SCHEMBL1058641 0.81 POLB (0.49) PDK1PDK2PDK3PDK4PSEN1
SCHEMBL8699830 0.81 POLB (0.49) PDK1PDK2PDK3PDK4PSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed