SCHEMBL7819795

SCHEMBL7819795

CC(=O)OCC(CCn1cnc2nc(N)nc(I)c21)COC(C)=O

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
HPGD P15428 1/20 0.57
ADRA1A P35348 1/20 0.57
HSD17B10 Q99714 1/20 0.57
RXFP1 Q9HBX9 1/20 0.57
ADORA2B P29275 1/20 0.34
CYP2C19 P33261 1/20 0.32
DUT P33316 1/20 0.32
P2RY1 P47900 2/20 0.31
TLR7 Q9NYK1 2/20 0.31
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3155510 0.88 KDM4E (0.58) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL7813547 0.82 KDM4E (0.66) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL7813412 0.80 KDM4E (0.48) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL7814812 0.80 ALDH1A1 (0.48) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL3158156 0.80 KDM4E (0.69) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL7981421 0.78 KDM4E (0.47) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL9873437 0.78 ALDH1A1 (0.46) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL7967624 0.77 KDM4E (0.46) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL14163777 0.75 KDM4E (0.69) KDM4EALDH1A1HPGDADRA1AHSD17B10
SCHEMBL3155583 0.74 KDM4E (0.67) KDM4EALDH1A1HPGDADRA1AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0352953-B1 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 2001-01-03 EP disclosed
US-5017701-A Process for the preparation of purine derivatives BEECHAM GROUP, P.L.C. (GB) 1991-05-21 US disclosed
EP-0352953-A2 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 1990-01-31 EP disclosed