SCHEMBL7814812

SCHEMBL7814812

CC(=O)OCC(CCn1cnc2nc(N)nc(SCc3ccc(C)cc3)c21)COC(C)=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
HPGD P15428 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ADRA1A P35348 1/20 0.48
HSD17B10 Q99714 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
CYP2C19 P33261 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
HIF1A Q16665 2/20 0.37
CYP2D6 P10635 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.36
TSHR P16473 1/20 0.36
RECQL P46063 1/20 0.36
GAA P10253 1/20 0.34
TP53 P04637 1/20 0.34
PHLPP2 Q6ZVD8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7816726 0.86 ALDH1A1 (0.55) ALDH1A1HPGDKDM4EADRA1AHSD17B10
SCHEMBL7813412 0.81 KDM4E (0.48) ALDH1A1HPGDKDM4EADRA1AHSD17B10
SCHEMBL9873437 0.80 ALDH1A1 (0.46) ALDH1A1HPGDKDM4EADRA1AHSD17B10
SCHEMBL7819795 0.80 KDM4E (0.57) ALDH1A1HPGDKDM4EADRA1AHSD17B10
SCHEMBL3155510 0.79 KDM4E (0.58) ALDH1A1HPGDKDM4EADRA1AHSD17B10
SCHEMBL7814637 0.78 CYP1A2 (0.59) ALDH1A1HPGDKDM4EADRA1AHSD17B10
SCHEMBL6317462 0.75 ALDH1A1 (0.56) ALDH1A1HPGDKDM4EADRA1AHSD17B10
SCHEMBL3158156 0.71 KDM4E (0.69) ALDH1A1HPGDKDM4EADRA1AHSD17B10
SCHEMBL7981421 0.70 KDM4E (0.47) ALDH1A1HPGDKDM4EADRA1AHSD17B10
SCHEMBL14163777 0.69 KDM4E (0.69) ALDH1A1HPGDKDM4EADRA1AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0352953-B1 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 2001-01-03 EP disclosed
US-5017701-A Process for the preparation of purine derivatives BEECHAM GROUP, P.L.C. (GB) 1991-05-21 US disclosed
EP-0352953-A2 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 1990-01-31 EP disclosed