SCHEMBL7819952

SCHEMBL7819952

CC(=O)Nc1nc2cc(-c3ccc4c(c3)CN(c3ncnc5c3CC(C)(C)CC5)CCO4)cnc2s1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PIK3CA P42336 10/20 0.36
PIK3CG P48736 6/20 0.35
PIK3CD O00329 3/20 0.33
PIK3CB P42338 3/20 0.33
OGA O60502 2/20 0.33
MTOR P42345 1/20 0.33
PIK3C3 Q8NEB9 1/20 0.33
CYP3A4 P08684 1/20 0.33
CREBBP Q92793 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7816149 0.89 PDE4B (0.34) PIK3CAPIK3CGPIK3CDPIK3CB
SCHEMBL858672 0.88 NPC1 (0.36) NPC1RAB9ASMN1; SMN2PIK3CAPIK3CG
SCHEMBL856936 0.87 PIK3CD (0.37) RAB9ASMN1; SMN2PIK3CAPIK3CGPIK3CD
SCHEMBL7816145 0.86 PIK3CA (0.34) PIK3CAPIK3CGPIK3CDPIK3CBMTOR
SCHEMBL858963 0.84 GPR142 (0.36) NPC1RAB9ASMN1; SMN2PIK3CAPIK3CG
SCHEMBL3758925 0.80 GPR142 (0.36) PIK3CACREBBP
SCHEMBL856291 0.80 USP2 (0.34) PIK3CAPIK3CGPIK3CDPIK3CBMTOR
SCHEMBL3758825 0.80 PDE10A (0.41) PIK3CAPIK3CGPIK3CDPIK3CBMTOR
SCHEMBL3716278 0.80 PIK3CA (0.40) PIK3CAPIK3CGCREBBP
SCHEMBL858091 0.79 PIK3CA (0.40) PIK3CAPIK3CGPIK3CDPIK3CBMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010135568-A1 BENZOXAZEPINES AS INHIBITORS OF MTOR AND THEIR USE TO TREAT CANCER EXELIXIS, INC. (US) 2010-11-25 WO disclosed