SCHEMBL7819985

SCHEMBL7819985

CN(C)CCn1nc2c3c(c(Cl)ccc31)C(=O)c1cccnc1-2

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 12/20 0.51
IDO1 P14902 3/20 0.39
TDO2 P48775 2/20 0.39
TDP2 O95551 1/20 0.38
NSD2 O96028 1/20 0.38
ABL1 P00519 1/20 0.38
PLCG1 P19174 1/20 0.38
CES1 P23141 1/20 0.38
PAX8 Q06710 1/20 0.38
RIN1 Q13671 1/20 0.38
GAA P10253 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
S100A4 P26447 1/20 0.36
CDC25B P30305 1/20 0.36
HTR6 P50406 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7816711 0.92 TOP2A (0.51) TOP2AIDO1TDO2TDP1S100A4
SCHEMBL7816428 0.84 TOP2A (0.45) TOP2AIDO1TDO2
SCHEMBL7809332 0.82 TDP2 (0.45) TOP2AIDO1TDP2NSD2ABL1
SCHEMBL7817109 0.81 TOP2A (0.44) TOP2AIDO1TDO2S100A4
SCHEMBL7804662 0.81 TOP2A (0.48) TOP2ATDP2TDP1CDC25B
SCHEMBL7819270 0.77 TOP2A (0.43) TOP2AIDO1TDO2
SCHEMBL10801094 0.77 TOP2A (0.46) TOP2A
SCHEMBL10799708 0.76 POLB (0.55) TOP2ANSD2
SCHEMBL7808475 0.76 TOP2A (0.47) TOP2AIDO1TDO2
SCHEMBL7812061 0.75 TOP2A (0.45) TOP2ATDP2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750619-B1 HETERO-ANNULATED INDAZOLES NOVUSPHARMA SPA (IT) 2001-05-30 EP disclosed
US-5596097-A ANTITUMOR AGENTS THE UNIVERSITY OF VERMONT (US) 1997-01-21 US disclosed
WO-1995024407-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1995-09-14 WO disclosed