SCHEMBL782091

SCHEMBL782091

COc1ccc(/C=C(\C#N)C(=O)O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.65
KDM4E B2RXH2 2/20 0.65
CYP3A4 P08684 2/20 0.65
HPGD P15428 2/20 0.65
CISD1 Q9NZ45 1/20 0.65
SLC16A3 O15427 1/20 0.65
SLC16A1 P53985 1/20 0.65
GPR35 Q9HC97 1/20 0.65
EGFR P00533 1/20 0.65
CYP1A2 P05177 1/20 0.62
MAPT P10636 1/20 0.62
TSHR P16473 1/20 0.62
NFKB1 P19838 1/20 0.62
APEX1 P27695 1/20 0.62
BLM P54132 1/20 0.62
PMP22 Q01453 1/20 0.62
NPSR1 Q6W5P4 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL782092 1.00 ALDH1A1 (0.65) ALDH1A1KDM4ECYP3A4HPGDCISD1
SCHEMBL4968638 1.00 ALDH1A1 (0.65) ALDH1A1KDM4ECYP3A4HPGDCISD1
SCHEMBL21625778 0.95 ALDH1A1 (0.59) ALDH1A1KDM4ECYP3A4HPGDCISD1
SCHEMBL21637629 0.95 ALDH1A1 (0.59) ALDH1A1KDM4ECYP3A4HPGDCISD1
SCHEMBL21625782 0.95 ALDH1A1 (0.59) ALDH1A1KDM4ECYP3A4HPGDCISD1
SCHEMBL7008415 0.88 SLC16A3 (0.57) ALDH1A1KDM4ECYP3A4HPGDCISD1
SCHEMBL28335121 0.88 SLC16A3 (0.67) ALDH1A1KDM4ECYP3A4HPGDCISD1
SCHEMBL17112792 0.88 KDM4E (0.64) ALDH1A1KDM4ECYP3A4HPGDCISD1
SCHEMBL17112791 0.88 KDM4E (0.64) ALDH1A1KDM4ECYP3A4HPGDCISD1
SCHEMBL13060202 0.88 MAPT (0.72) ALDH1A1KDM4ECYP3A4HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 162 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379625-B1 UV AND LIGHT PROTECTIVE FILM HUHTAMAKI FORCHHEIM (DE) 2013-02-20 EP claimed
EP-2379625-A1 UV AND LIGHT PROTECTIVE FILM Huhtamaki Forchheim Zweigniederlassung der Huhtamaki Deutschland GmbH & Co. KG (DE) 2011-10-26 EP claimed
US-20110083765-A1 UV LIGHT AND PROTECTIVE FILM HUHTAMAKI FORCHHEIM, ZWEIGNIEDERLASSUNG DER HUHTAMAKI DEUTSCHLAND GMBH & CO (DE) 2011-04-14 US claimed
WO-2010075946-A1 UV AND LIGHT PROTECTIVE FILM HUHTAMAKI FORCHHEIM, ZWEIGNIEDERLASSUNG DER HUHTAMAKI DEUTSCHLAND GMBH & CO. KG (DE) 2010-07-08 WO claimed
US-20040038234-A1 Sample generation for genotyping by mass spectrometry CONSORTIUM NATIONAL DE RECHERCHE EN GENOMIQUE (FR) 2004-02-26 US claimed
EP-1297181-A2 SAMPLE GENERATION FOR GENOTYPING BY MASS SPECTROMETRY Centre National de Genotype (FR) 2003-04-02 EP claimed
US-20020131939-A1 Hair protection compositions ROCHE VITAMINS INC. 2002-09-19 US claimed
EP-1036202-B1 METHOD FOR IDENTIFYING NUCLEIC ACIDS BY MEANS OF MATRIX-ASSISTED LASER DESORPTION/IONISATION MASS SPECTROMETRY MAX PLANCK GESELLSCHAFT (DE) 2002-05-02 EP claimed
EP-1170379-A1 Sample generation for genotyping by mass spectrometry Centre National de Genotypage (FR) 2002-01-09 EP claimed
WO-2002000931-A2 SAMPLE GENERATION FOR GENOTYPING BY MASS SPECTROMETRY CENTRE NATIONAL DE GENOTYPAGE (FR) 2002-01-03 WO claimed
EP-1036202-A2 METHOD FOR IDENTIFYING NUCLEIC ACIDS BY MEANS OF MATRIX-ASSISTED LASER DESORPTION/IONISATION MASS SPECTROMETRY MAX-PLANCK-GESELLSCHAFT ZUR FÖRDERUNG DER WISSENSCHAFTEN E.V. (DE) 2000-09-20 EP claimed
WO-1999029898-A2 METHOD FOR IDENTIFYING NUCLEIC ACIDS BY MEANS OF MATRIX-ASSISTED LASER DESORPTION/IONISATION MASS SPECTROMETRY MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 1999-06-17 WO claimed
EP-0713383-B1 SUNSCREEN AGENTS UNILEVER PLC (GB) 1998-06-17 EP claimed
US-5567418-A ADDING A /4-METHOXYBENZYLIDENE/CYANOACETATE/ L'OREAL (FR) 1996-10-22 US claimed
US-5538716-A SUNSCREEN AGENTS FOR SUNTAN LOTION L'OREAL (FR) 1996-07-23 US claimed
EP-0557089-B1 Sunscreen agents containing layered double hydroxides UNILEVER PLC (GB) 1996-05-29 EP claimed
EP-0551510-B1 PHOTOSTABLE FILTERING COSMETIC COMPOSITION CONTAINING A UV-A FILTER AND A 4-METHOXY BENZYLIDENE CYANOACETATE OREAL (FR) 1995-09-27 EP claimed
EP-0403238-A2 Cosmetic composition UNILEVER PLC (GB) 1990-12-19 EP claimed
US-4284621-A SUNSCREEN FOR SKIN BAYER AKTIENGESELLSCHAFT (DE) 1981-08-18 US claimed
EP-0005182-B1 COMPOSITION AGAINST THE ACTION OF LIGHT BAYER AG (DE) 1981-07-29 EP claimed