SCHEMBL7821052

SCHEMBL7821052

COc1ccc2nc(CCCCCCC(=O)O)ccc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 1/20 0.51
CYSLTR2 Q9NS75 4/20 0.50
CYSLTR1 Q9Y271 4/20 0.50
CYP1A2 P05177 3/20 0.49
CYP2C19 P33261 2/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CYP2E1 P05181 1/20 0.47
CYP2C8 P10632 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2B6 P20813 1/20 0.47
KDM4E B2RXH2 2/20 0.47
NPC1 O15118 1/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
MAOA P21397 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7829813 0.86 HDAC1 (0.56) HDAC1HDAC2HDAC3HDAC4HDAC7
Iodide SCHEMBL28230532 0.81 PDE10A (0.49) LTB4RCYSLTR2CYSLTR1CYP1A2CYP2C19
SCHEMBL5928217 0.80 NCF1 (0.54) CYP1A2CYP2C19ALDH1A1CYP2E1CYP2C8
SCHEMBL7831703 0.76 CYSLTR1 (0.64) LTB4RCYSLTR2CYSLTR1CYP1A2MAPT
SCHEMBL8649122 0.76 CYSLTR1 (0.64) LTB4RCYSLTR2CYSLTR1CYP1A2MAPT
SCHEMBL14127808 0.76 NCF1 (0.56) CYP1A2CYP2C19ALDH1A1HPGDCYP2E1
SCHEMBL9119048 0.76 KDM4E (0.48) CYP1A2ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL14352239 0.75 NCF1 (0.58) CYP1A2CYP2C19ALDH1A1CYP2E1CYP2C8
SCHEMBL9952773 0.75 CYSLTR1 (0.66) LTB4RCYSLTR2CYSLTR1CYP1A2MAPT
SCHEMBL27596905 0.75 NCF1 (0.54) CYP1A2CYP2C19ALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737671-B1 Aromatic hydroxamic acid compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-12-12 EP disclosed
US-5804601-A USEFUL FOR TREATING ALZHEIMER'S DISEASE, MULTIPLE SCLEROSIS, BACTERIAL OR VIRAL MENINGITIS, DOWN'S SYNDROME AND PARKINSON'S DISEASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-08 US disclosed
EP-0737671-A2 Aromatic hydroxamic acid compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1996-10-16 EP disclosed