SCHEMBL9119048

SCHEMBL9119048

COc1ccc2nc(CCC(=O)OC(C)(C)C)ccc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.48
NPC1 O15118 4/20 0.48
RAB9A P51151 4/20 0.48
HDAC1 Q13547 2/20 0.47
HDAC2 Q92769 2/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 2/20 0.46
LMNA P02545 2/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAOA P21397 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A3 Q01959 1/20 0.46
PDE10A Q9Y233 2/20 0.45
ALDH1A1 P00352 7/20 0.44
HPGD P15428 6/20 0.44
NCF1 P14598 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4548369 0.80 MAPT (0.67) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL7821052 0.76 LTB4R (0.51) KDM4ENPC1RAB9AHDAC1HDAC2
SCHEMBL14127808 0.75 NCF1 (0.56) KDM4ENPC1RAB9AHDAC1HDAC2
SCHEMBL24744929 0.75 KDM4E (0.52) KDM4ENPC1RAB9AHDAC1HDAC2
SCHEMBL7453174 0.75 POLB (0.40) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL7453167 0.75 POLB (0.40) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL27596905 0.74 NCF1 (0.54) KDM4ENPC1RAB9AHDAC1HDAC2
SCHEMBL14352239 0.74 NCF1 (0.58) KDM4ENPC1RAB9AHDAC1HDAC2
SCHEMBL14094660 0.74 NCF1 (0.54) KDM4ENPC1RAB9AHDAC1HDAC2
SCHEMBL7808259 0.73 NCF1 (0.57) KDM4ENPC1RAB9AHDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434186-A Antiinflammatory agents HOFFMANN-LA ROCHE INC. (US) 1995-07-18 US disclosed
US-5273999-A A 4-keto-boroalkyleneoxychroman or 2,3-dihydrobenzofuran derivative HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
EP-0531823-A1 Bicyclic carboxylic acid derivatives as anti-inflammatory agents F. HOFFMANN-LA ROCHE AG (CH) 1993-03-17 EP disclosed