SCHEMBL7822004

SCHEMBL7822004

COc1ccc(-c2cc3cc4c(cc3c(C)n2)OCO4)cc1OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.60
MAPT P10636 3/20 0.60
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
RAC1 P63000 4/20 0.54
TOP2A P11388 1/20 0.54
IDO1 P14902 1/20 0.52
TDO2 P48775 1/20 0.52
ALDH1A1 P00352 3/20 0.49
GAA P10253 1/20 0.49
KIT P10721 1/20 0.48
FLT3 P36888 1/20 0.47
CASP3 P42574 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
TSHR P16473 2/20 0.46
MAPK1 P28482 2/20 0.46
USP2 O75604 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3318529 0.87 KDM4E (0.64) KDM4EMAPTNPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL3316173 0.86 KDM4E (0.62) KDM4EMAPTNPC1RAB9AMEN1
SCHEMBL7822956 0.83 KDM4E (0.83) KDM4EMAPTNPC1RAB9AMEN1
SCHEMBL9679340 0.76 NPC1 (0.58) KDM4EMAPTNPC1RAB9AMEN1
SCHEMBL3321436 0.73 RAC1 (0.84) KDM4EMAPTNPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL3318470 0.72 RAC1 (0.85) KDM4EMAPTNPC1RAB9AMEN1
SCHEMBL3321880 0.72 KDM4E (0.80) KDM4EMAPTNPC1RAB9AMEN1
SCHEMBL15436211 0.71 KIT (0.58) KDM4EMAPTNPC1RAB9AMEN1
SCHEMBL29365587 0.71 ALOX5 (0.72) KDM4EMAPTMEN1KMT2ATOP2A
SCHEMBL3324961 0.71 KDM4E (1.00) KDM4EMAPTNPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888346-B1 CORALYNE ANALOGS AS TOPOISOMERASE INHIBITORS UNIV RUTGERS (US) 2001-06-06 EP disclosed
EP-0888346-A1 CORALYNE ANALOGS AS TOPOISOMERASE INHIBITORS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 1999-01-07 EP disclosed
WO-1997029106-A1 CORALYNE ANALOGS AS TOPOISOMERASE INHIBITORS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 1997-08-14 WO disclosed