SCHEMBL7823682

SCHEMBL7823682

Cc1nc2cccc(CBr)c2c(=O)n1COCC[Si](C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ELANE P08246 8/20 0.45
NPC1 O15118 1/20 0.36
KCNH2 Q12809 5/20 0.35
HRH3 Q9Y5N1 5/20 0.35
TSHR P16473 2/20 0.33
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7815551 0.86 HRH3 (0.43) ELANENPC1KCNH2HRH3
SCHEMBL5369563 0.85 ELANE (0.42) ELANENPC1
SCHEMBL4932747 0.84 ELANE (0.43) ELANENPC1TSHRHSD17B10MEN1
SCHEMBL7827132 0.82 HDAC1 (0.37) ELANENPC1KCNH2HRH3TSHR
SCHEMBL7823078 0.79 PARP1 (0.38) NPC1TSHRMEN1KMT2A
SCHEMBL7822854 0.78 NPC1 (0.42) NPC1TSHRMEN1KMT2A
SCHEMBL23209066 0.77 AKR1B10 (0.34) NPC1HSD17B10MEN1KMT2A
SCHEMBL29970272 0.77 AKR1B10 (0.34) NPC1HSD17B10MEN1KMT2A
SCHEMBL1542331 0.73 NPC1 (0.36) ELANENPC1KMT2A
SCHEMBL29991937 0.72 ATM (0.47) NPC1HSD17B10MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0637300-B1 ANTIPROLIFERATIVE QUINAZOLINES AGOURON PHARMA (US) 2001-09-05 EP disclosed
US-5885996-A AN ENZYME INHIBITORS OF THYMIDYLATE SYNTHASE WORKS AS BACTERICIDES, FUNGICIDES INHIBITING YEASTS, FUNGI AGOURON PHARMACEUTICALS, INC. (US) 1999-03-23 US disclosed
US-5707992-A MICROBIOCIDES, ANTITUMOR AGENTS AGOURON PHARMACEUTICALS, INC. (US) 1998-01-13 US disclosed
US-5430148-A Antiproliferative quinazolines AGOURON PHARMACEUTICALS, INC. (US) 1995-07-04 US disclosed
EP-0637300-A1 ANTIPROLIFERATIVE QUINAZOLINES AGOURON PHARMACEUTICALS, INC. (US) 1995-02-08 EP disclosed
WO-1993020055-A1 ANTIPROLIFERATIVE QUINAZOLINES AGOURON PHARMACEUTICALS, INC. (US) 1993-10-14 WO disclosed