SCHEMBL7824409

SCHEMBL7824409

CCOC(=O)CNc1ccc(C)c(C)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.56
ALDH1A1 P00352 5/20 0.50
LMNA P02545 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
IDH1 O75874 2/20 0.46
MAPT P10636 5/20 0.46
HTT P42858 2/20 0.46
DHODH Q02127 2/20 0.46
KDM4E B2RXH2 2/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
EGFR P00533 1/20 0.44
GAA P10253 1/20 0.43
USP2 O75604 1/20 0.43
TSHR P16473 1/20 0.43
RECQL P46063 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3142563 0.87 POLB (0.54) POLBLMNATDP1IDH1HTT
SCHEMBL5113179 0.86 POLB (0.53) POLBALDH1A1LMNATDP1MAPT
SCHEMBL28658507 0.86 POLB (0.52) POLBALDH1A1LMNATDP1IDH1
Hydrochloric Acid SCHEMBL5775146 0.85 POLB (0.51) POLBALDH1A1LMNATDP1MAPT
SCHEMBL9830208 0.84 ALDH1A1 (0.51) POLBALDH1A1LMNAMAPTHTT
SCHEMBL11355645 0.83 POLB (0.55) POLBALDH1A1LMNAIDH1MAPT
SCHEMBL11471191 0.82 POLB (0.48) POLBALDH1A1LMNATDP1MAPT
SCHEMBL6906565 0.82 POLB (0.55) POLBLMNATDP1IDH1HTT
SCHEMBL29148948 0.81 POLB (0.61) POLBLMNAIDH1MAPTHTT
SCHEMBL4035087 0.81 POLB (0.65) POLBALDH1A1TDP1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117447339-A Method for preparing alkyl substituted glycine derivative by driving visible light 沈阳师范大学 2024-01-26 CN disclosed
EP-3560928-B1 FUSED IMIDAZOLE COMPOUND HAVING INDOLEAMINE 2,3-DIOXYGENASE INHIBITORY ACTIVITY SHENZHEN CHIPSCREEN BIOSCIENCES CO LTD (CN) 2021-10-20 EP disclosed
CN-108203438-B Fused imidazole compounds having indoleamine 2,3-dioxygenase inhibitory activity 深圳微芯生物科技股份有限公司 2021-09-28 CN disclosed
US-10604529-B2 Fused imidazole compound having indoleamine 2,3-dioxygenase inhibitory activity SHENZHEN CHIPSCREEN BIOSCIENCES CO., LTD. (CN) 2020-03-31 US disclosed
US-20190352307-A1 FUSED IMIDAZOLE COMPOUND HAVING INDOLEAMINE 2,3-DIOXYGENASE INHIBITORY ACTIVITY SHENZHEN CHIPSCREEN BIOSCIENCES CO., LTD. (CN) 2019-11-21 US disclosed
EP-3560928-A1 FUSED IMIDAZOLE COMPOUND HAVING INDOLEAMINE 2,3-DIOXYGENASE INHIBITORY ACTIVITY Shenzhen Chipscreen Biosciences Co., Ltd. (CN) 2019-10-30 EP disclosed
WO-2018113624-A1 FUSED IMIDAZOLE COMPOUND HAVING INDOLEAMINE 2,3-DIOXYGENASE INHIBITORY ACTIVITY 深圳微芯生物科技有限责任公司 2018-06-28 WO disclosed
EP-0721944-B1 IMIDAZOLIDINE DERIVATIVE AND USE THEREOF SUNTORY LTD (JP) 2001-01-17 EP disclosed
US-5691335-A CARDIOVASCULAR DISORDERS SUNTORY LIMITED (JP) 1997-11-25 US disclosed
EP-0721944-A1 IMIDAZOLIDINE DERIVATIVE AND USE THEREOF SUNTORY LIMITED (JP) 1996-07-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190352307-A1 FUSED IMIDAZOLE COMPOUND HAVING INDOLEAMINE 2,3-DIOXYGENASE INHIBITORY ACTIVITY IDO1, IDO2, INMT POLB 3522/4885ALDH1A1 735/4885LMNA 4703/4885
US-10604529-B2 Fused imidazole compound having indoleamine 2,3-dioxygenase inhibitory activity IDO1, IDO2, INMT POLB 3731/4885ALDH1A1 376/4885LMNA 4738/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.