SCHEMBL7825628

SCHEMBL7825628

CCc1ccc2c(=O)c3[nH]nnc3c(=O)[nH]c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 6/20 0.46
CYP2C9 P11712 3/20 0.46
KIF11 P52732 1/20 0.42
DAO P14920 1/20 0.42
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CDK2 P24941 2/20 0.35
CCNE2 O96020 1/20 0.35
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
CCNE1 P24864 1/20 0.35
TYMS P04818 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
CDK1 P06493 1/20 0.34
PDE9A O76083 1/20 0.34
MAOA P21397 1/20 0.33
DYRK1A Q13627 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7826505 0.90 PTGES (0.47) PTGESCYP2C9DAOALDH1A1MAOA
SCHEMBL7826259 0.86 PTGES (0.51) PTGESCYP2C9KDM4ENPC1ALDH1A1
SCHEMBL7815632 0.85 PARP1 (0.50) PTGESCYP2C9KDM4ENPC1RAB9A
SCHEMBL7822908 0.83 KDM4E (0.38) PTGESCYP2C9KDM4ENPC1ALDH1A1
SCHEMBL7827947 0.82 PTGES (0.43) PTGESKIF11DAOKDM4ENPC1
SCHEMBL7830520 0.82 HSP90AA1 (0.39) PTGESCYP2C9KDM4EALDH1A1MEN1
SCHEMBL7815301 0.82 KDM4E (0.42) KDM4ENPC1ALDH1A1RAB9AMAOA
SCHEMBL7827211 0.81 HSD17B10 (0.51) KDM4ENPC1ALDH1A1CDK2CCNE2
SCHEMBL7824009 0.81 PARP1 (0.46) PTGESCYP2C9KDM4EALDH1A1
SCHEMBL7830466 0.81 PARP1 (0.39) KDM4EALDH1A1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686636-B1 TRICYCLIC BENZAZEPINE AND BENZOTHIAZEPINE DERIVATIVES MEIJI SEIKA CO (JP) 2001-04-04 EP disclosed
EP-0686636-A1 TRICYCLIC BENZAZEPINE AND BENZOTHIAZEPINE DERIVATIVES MEIJI SEIKA KABUSHIKI KAISHA (JP) 1995-12-13 EP disclosed