SCHEMBL7826372

SCHEMBL7826372

CCc1cc(OC[C@@H]2CCN2C)cnc1F

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 8/20 0.55
CHRNA4 P43681 7/20 0.55
CHRNA3 P32297 4/20 0.53
DAPK3 O43293 1/20 0.52
ROCK2 O75116 1/20 0.52
PRKCG P05129 1/20 0.52
PIM1 P11309 1/20 0.52
RPS6KB1 P23443 1/20 0.52
AKT1 P31749 1/20 0.52
LIMK1 P53667 1/20 0.52
CDK5 Q00535 1/20 0.52
PRKCD Q05655 1/20 0.52
PAK1 Q13153 1/20 0.52
STK3 Q13188 1/20 0.52
ROCK1 Q13464 1/20 0.52
DYRK1A Q13627 1/20 0.52
CDC42BPA Q5VT25 1/20 0.52
PRKD2 Q9BZL6 1/20 0.52
IRAK4 Q9NWZ3 1/20 0.52
CHRNB4 P30926 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7824581 1.00 CHRNB2 (0.55) CHRNB2CHRNA4CHRNA3DAPK3ROCK2
SCHEMBL7826660 0.92 CHRNB2 (0.66) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1
SCHEMBL7828958 0.92 CHRNB2 (0.66) CHRNB2CHRNA4CHRNA3CHRNB4CHRNB1
SCHEMBL7408434 0.86 CHRNB2 (0.48) CHRNB2CHRNA4CHRNA3DAPK3ROCK2
SCHEMBL7410484 0.86 CHRNB2 (0.48) CHRNB2CHRNA4CHRNA3DAPK3ROCK2
SCHEMBL7823561 0.85 CHRNA3 (0.54) CHRNB2CHRNA4CHRNA3DAPK3ROCK2
SCHEMBL7817925 0.85 CHRNA3 (0.54) CHRNB2CHRNA4CHRNA3DAPK3ROCK2
SCHEMBL7827624 0.84 CHRNA3 (0.56) CHRNB2CHRNA4CHRNA3DAPK3ROCK2
SCHEMBL7825999 0.84 CHRNA3 (0.56) CHRNB2CHRNA4CHRNA3DAPK3ROCK2
SCHEMBL7827635 0.83 CHRNA3 (0.52) CHRNB2CHRNA4CHRNA3DAPK3ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0846114-B1 3-PYRIDYLOXYALKYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LAB (US) 2001-12-05 EP claimed
EP-0846114-B1 3-PYRIDYLOXYALKYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LAB (US) 2001-12-05 EP disclosed