SCHEMBL7827697

SCHEMBL7827697

COC(=O)c1c(N)ccc(C)c1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.42
HSD17B10 Q99714 4/20 0.42
CFTR P13569 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
PRKCZ Q05513 2/20 0.41
HPGD P15428 5/20 0.40
MAPT P10636 4/20 0.40
GAA P10253 4/20 0.40
KDM4E B2RXH2 4/20 0.40
TSHR P16473 2/20 0.40
ALOX15 P16050 1/20 0.40
RAB9A P51151 1/20 0.40
CYP3A4 P08684 2/20 0.40
ACHE P22303 1/20 0.40
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL773070 0.83 ALDH1A1 (0.46) ALDH1A1HSD17B10CFTRCA12CA1
SCHEMBL7461675 0.81 ALDH1A1 (0.44) ALDH1A1HSD17B10CFTRCA12CA1
SCHEMBL8178102 0.81 ALDH1A1 (0.41) ALDH1A1HSD17B10CFTRCA12CA1
SCHEMBL29284888 0.80 CA12 (0.57) ALDH1A1HSD17B10CA12CA1CA2
SCHEMBL3104246 0.79 KDM4E (0.41) ALDH1A1MAPTKDM4ETSHRCYP3A4
SCHEMBL1335494 0.79 GRM6 (0.42) ALDH1A1HSD17B10CFTRCA12CA1
SCHEMBL3530996 0.79 ALDH1A1 (0.42) ALDH1A1HSD17B10CFTRCA12CA1
SCHEMBL27474595 0.79 ABL1 (0.45) ALDH1A1HSD17B10CFTRCA12CA1
SCHEMBL9447396 0.79 GRM6 (0.42) ALDH1A1HSD17B10CFTRCA12CA1
SCHEMBL16096788 0.79 NCEH1 (0.42) ALDH1A1HSD17B10CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1335307-A Synthesis process of 2-amino quinbolone compounds MILITARY MEDICAL UNIV NO 1 PLA (CN) 2002-02-13 CN disclosed
EP-0637300-B1 ANTIPROLIFERATIVE QUINAZOLINES AGOURON PHARMA (US) 2001-09-05 EP disclosed
EP-0637300-A1 ANTIPROLIFERATIVE QUINAZOLINES AGOURON PHARMACEUTICALS, INC. (US) 1995-02-08 EP disclosed
WO-1993020055-A1 ANTIPROLIFERATIVE QUINAZOLINES AGOURON PHARMACEUTICALS, INC. (US) 1993-10-14 WO disclosed