SCHEMBL7828344

SCHEMBL7828344

CN1CCc2ccc(N=C(N)c3cccs3)cc2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 15/20 1.00
NOS1 P29475 18/20 0.65
NOS2 P35228 14/20 0.65
CHRM2 P08172 1/20 0.55
ADRA2A P08913 1/20 0.55
CYP2D6 P10635 1/20 0.55
CHRM1 P11229 1/20 0.55
ADRA2B P18089 1/20 0.55
ADRA2C P18825 1/20 0.55
CHRM3 P20309 1/20 0.55
ADRA1D P25100 1/20 0.55
HTR1B P28222 1/20 0.55
ADRA1A P35348 1/20 0.55
ADRA1B P35368 1/20 0.55
KCNH2 Q12809 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7827939 0.99 NOS3 (0.98) NOS3NOS1NOS2
SCHEMBL7817523 0.87 NOS3 (0.76) NOS3NOS1NOS2KCNH2
SCHEMBL7826140 0.86 NOS3 (0.76) NOS3NOS1NOS2KCNH2
SCHEMBL7817443 0.86 NOS3 (0.76) NOS3NOS1NOS2CHRM2ADRA2A
Hydrochloric Acid SCHEMBL7828295 0.86 NOS3 (0.74) NOS3NOS1NOS2KCNH2
Hydrochloric Acid SCHEMBL7832875 0.85 NOS3 (0.74) NOS3NOS1NOS2KCNH2
SCHEMBL7511366 0.85 NOS3 (0.74) NOS3NOS1NOS2KCNH2
SCHEMBL7824443 0.85 NOS3 (0.73) NOS3NOS1NOS2KCNH2
Hydrochloric Acid SCHEMBL7510751 0.84 NOS3 (0.72) NOS3NOS1NOS2KCNH2
SCHEMBL7482097 0.83 NOS3 (0.71) NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0983266-B1 novel tetrahydroisoquinolin thiophenecarboximidamides ASTRAZENECA AB (SE) 2001-12-12 EP claimed
EP-0983266-A1 COMPOUNDS Astra Aktiebolag (SE) 2000-03-08 EP claimed
WO-1998050380-A1 COMPOUNDS ASTRA AKTIEBOLAG (SE) 1998-11-12 WO claimed
EP-0983266-B1 novel tetrahydroisoquinolin thiophenecarboximidamides ASTRAZENECA AB (SE) 2001-12-12 EP disclosed
US-6166030-A Compounds ASTRA AKTIEBOLAG (SE) 2000-12-26 US disclosed
EP-0983266-A1 COMPOUNDS Astra Aktiebolag (SE) 2000-03-08 EP disclosed
WO-1998050380-A1 COMPOUNDS ASTRA AKTIEBOLAG (SE) 1998-11-12 WO disclosed