SCHEMBL7828544

SCHEMBL7828544

c1cc(-n2ccnc2)cc(-n2cnc3cc(-c4ccco4)ccc32)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
RAB9A P51151 5/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
NPC1 O15118 4/20 0.42
KDM4E B2RXH2 4/20 0.42
MAPT P10636 3/20 0.42
GAA P10253 2/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 3/20 0.41
TP53 P04637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
IDO1 P14902 1/20 0.40
KDR P35968 2/20 0.39
NCOA3 Q9Y6Q9 1/20 0.38
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
CYP3A4 P08684 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7832246 0.89 ALDH1A1 (0.42) ALDH1A1RAB9ASMN1; SMN2NPC1KDM4E
SCHEMBL2643078 0.83 CYP3A4 (0.49) ALDH1A1RAB9ASMN1; SMN2NPC1KDM4E
SCHEMBL2646699 0.83 KDR (0.54) ALDH1A1RAB9ASMN1; SMN2NPC1KDM4E
SCHEMBL2643461 0.82 IDO1 (0.40) ALDH1A1RAB9ASMN1; SMN2NPC1KDM4E
SCHEMBL2646102 0.80 GABRA1 (0.52) ALDH1A1RAB9ASMN1; SMN2NPC1KDM4E
SCHEMBL2656192 0.80 IDO1 (0.49) ALDH1A1RAB9ASMN1; SMN2NPC1KDM4E
SCHEMBL2643844 0.78 GRM5 (0.53) ALDH1A1RAB9ASMN1; SMN2NPC1KDM4E
SCHEMBL2647252 0.78 FGFR1 (0.62) ALDH1A1RAB9ASMN1; SMN2NPC1HPGD
SCHEMBL20510883 0.77 FGFR1 (0.58) IDO1CYP3A4HTTFGFR1
SCHEMBL7819811 0.76 FGFR1 (0.41) ALDH1A1RAB9ASMN1; SMN2NPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1164134-A1 Benzimidazole compounds and their use as modulators of the GABA A receptor complex NEUROSEARCH A/S (DK) 2001-12-19 EP claimed
US-5922724-A Benzimidazole compounds and their use as modulators of the GABA a receptor complex NEUROSEARCH A/S (DK) 1999-07-13 US claimed
EP-1164134-A1 Benzimidazole compounds and their use as modulators of the GABA A receptor complex NEUROSEARCH A/S (DK) 2001-12-19 EP disclosed
US-5922724-A Benzimidazole compounds and their use as modulators of the GABA a receptor complex NEUROSEARCH A/S (DK) 1999-07-13 US disclosed