SCHEMBL7828564

SCHEMBL7828564

NCCCNc1cccc(-c2ccc(-c3ccccc3)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.48
ALDH1A1 P00352 1/20 0.48
NPY1R P25929 1/20 0.48
NPY5R Q15761 1/20 0.48
MGLL Q99685 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.43
TAAR1 Q96RJ0 3/20 0.42
HDAC6 Q9UBN7 5/20 0.42
HDAC1 Q13547 4/20 0.42
SYK P43405 2/20 0.41
CFD P00746 2/20 0.41
HDAC3 O15379 2/20 0.40
HDAC4 P56524 2/20 0.40
HDAC7 Q8WUI4 2/20 0.40
HDAC2 Q92769 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22631193 0.83 MAPT (0.54) MAPTALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL7838920 0.82 PRKCA (0.40) MAPTALDH1A1NPY1RNPY5RHTT
SCHEMBL1072934 0.81 MAPT (0.73) MAPTALDH1A1HDAC1HDAC3HDAC2
SCHEMBL14149699 0.81 MAPT (0.50) MAPTALDH1A1MGLLCYP1A2CYP3A4
SCHEMBL30505169 0.81 MAPT (0.50) MAPTALDH1A1MGLLCYP1A2CYP3A4
SCHEMBL28653602 0.81 ALDH1A1 (0.50) MAPTALDH1A1MGLLHDAC6HDAC1
Hydrochloric Acid SCHEMBL12477885 0.79 ALDH1A1 (0.70) MAPTALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL11935615 0.79 ALDH1A1 (0.52) MAPTALDH1A1NPY1RNPY5RTAAR1
SCHEMBL11934955 0.79 ALDH1A1 (0.52) MAPTALDH1A1NPY1RNPY5RTAAR1
SCHEMBL11253095 0.77 MAPT (0.46) MAPTALDH1A1MGLLCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144381-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GmbH (DE) 2001-10-17 EP disclosed
WO-2000032577-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GMBH (DE) 2000-06-08 WO disclosed