SCHEMBL7830706

SCHEMBL7830706

COc1cccc(OC)c1OCc1nc2cc(-n3ccnc3)ccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.46
RAB9A P51151 5/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
MAOA P21397 2/20 0.46
MAOB P27338 2/20 0.46
CYP11B1 P15538 3/20 0.43
CYP11B2 P19099 3/20 0.43
TP53 P04637 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
CBFB Q13951 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.40
CYP19A1 P11511 2/20 0.40
F9 P00740 1/20 0.40
CYP1A2 P05177 3/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2D6 P10635 3/20 0.38
CYP2C19 P33261 2/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7821793 0.99 NPC1 (0.46) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7833671 0.94 NPC1 (0.43) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7837220 0.93 NPC1 (0.43) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7834952 0.93 MAOA (0.42) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7830709 0.92 CBFB (0.50) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7834944 0.92 MAOA (0.41) NPC1RAB9ASMN1; SMN2MAOAMAOB
Hydrochloric Acid SCHEMBL7821802 0.91 CBFB (0.49) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7832658 0.91 NPC1 (0.40) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7830427 0.91 CYP11B1 (0.47) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7832653 0.88 F9 (0.44) NPC1RAB9ASMN1; SMN2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894795-B1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-06 EP claimed
EP-0894795-A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-02-03 EP claimed
EP-0894795-B1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-06 EP disclosed
EP-0894795-A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-02-03 EP disclosed