SCHEMBL7833671

SCHEMBL7833671

COc1cccc(C)c1OCc1nc2cc(-n3ccnc3)ccc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.43
RAB9A P51151 6/20 0.43
SMN1; SMN2 Q16637 5/20 0.43
MAOA P21397 2/20 0.43
MAOB P27338 2/20 0.43
F9 P00740 1/20 0.41
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
TP53 P04637 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
CBFB Q13951 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
CYP19A1 P11511 1/20 0.37
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7830706 0.94 NPC1 (0.46) NPC1RAB9ASMN1; SMN2MAOAMAOB
Hydrochloric Acid SCHEMBL7821793 0.93 NPC1 (0.46) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7833677 0.93 CBFB (0.47) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7832653 0.92 F9 (0.44) NPC1RAB9ASMN1; SMN2F9CYP11B1
Hydrochloric Acid SCHEMBL8155873 0.91 F9 (0.44) NPC1RAB9ASMN1; SMN2F9CYP11B1
SCHEMBL7837220 0.90 NPC1 (0.43) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7834952 0.89 MAOA (0.42) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7834944 0.88 MAOA (0.41) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7830709 0.86 CBFB (0.50) NPC1RAB9ASMN1; SMN2MAOAMAOB
SCHEMBL7830427 0.85 CYP11B1 (0.47) NPC1RAB9ASMN1; SMN2MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894795-B1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-06 EP disclosed
US-6040327-A INHIBITORS OF INTERLEUKINS; TREATING RHEUMATOID ARTHRITIS OR ARTHROSIS ADIR ET COMPAGNIE (FR) 2000-03-21 US disclosed
EP-0894795-A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-02-03 EP disclosed