SCHEMBL7830810

SCHEMBL7830810

CC(=O)OC(C(N)=O)c1cccc(-c2nccs2)c1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNB1 Q14721 8/20 0.44
KCNA5 P22460 1/20 0.43
CTSA P10619 7/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.41
LRRK2 Q5S007 1/20 0.41
FFAR1 O14842 1/20 0.40
PDPK1 O15530 1/20 0.40
KAT6A Q92794 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6216984 0.76 CYP1A2 (0.47) KCNB1KCNA5CTSAPTGDR2LRRK2
SCHEMBL13801391 0.76 PDPK1 (0.55) KCNB1KCNA5CTSAPDPK1
SCHEMBL28405984 0.74 PDPK1 (0.51) KCNB1KCNA5CTSAPDPK1
SCHEMBL5888543 0.74 PDPK1 (0.51) KCNB1KCNA5CTSAPDPK1
SCHEMBL29793545 0.74 PDPK1 (0.51) KCNB1KCNA5CTSAPDPK1
SCHEMBL28866312 0.72 KCNB1 (0.46) KCNB1KCNA5CTSAPTGDR2LRRK2
SCHEMBL31079263 0.72 ALDH1A1 (0.41) CTSA
SCHEMBL20545939 0.72 CTSA (0.57) CTSAPTGDR2
SCHEMBL20545938 0.72 CTSA (0.57) CTSAPTGDR2
SCHEMBL30671345 0.71 KCNB1 (0.51) KCNB1KCNA5CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1124810-A1 2-AMINO-THIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2001-08-22 EP disclosed
WO-2000026202-A1 2-AMINO-THIAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-05-11 WO disclosed