SCHEMBL7830820

SCHEMBL7830820

Nc1nc(-c2ccc3c(c2)CC(=O)N3)nc2[nH]cnc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
GRIA1 P42261 5/20 0.45
CACNG8 Q8WXS5 2/20 0.44
CRBN Q96SW2 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
PGR P06401 3/20 0.41
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
NEK2 P51955 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7833215 0.99 PDE3B (0.46) PDE3BPDE3AGRIA1CACNG8CRBN
SCHEMBL7830814 0.81 NEK2 (0.48) PDE3BPDE3AGRIA1CACNG8CYP1A2
Hydrochloric Acid SCHEMBL7833212 0.81 NEK2 (0.48) PDE3BPDE3AGRIA1CACNG8CYP1A2
SCHEMBL7821784 0.77 ALDH1A1 (0.42) CYP11B1CYP11B2ALDH1A1MAPTHTT
SCHEMBL15756771 0.70 DPP4 (0.41) POLBSMN1; SMN2
SCHEMBL1741363 0.70 ADORA2A (0.46) POLBHTT
SCHEMBL17815691 0.70 RIPK1 (0.44)
SCHEMBL10711906 0.69 PDE3B (0.68) PDE3BPDE3AGRIA1CACNG8CRBN
SCHEMBL10659225 0.69 MAPT (0.78) PDE3BPDE3AGRIA1CACNG8CYP1A2
SCHEMBL7249955 0.69 IDO1 (0.43) ALDH1A1MAPTHTTSMN1; SMN2AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP claimed
EP-0802914-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.p.A. (IT) 1997-10-29 EP claimed
WO-1997018212-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.P.A. (IT) 1997-05-22 WO claimed
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP disclosed