SCHEMBL7830973

SCHEMBL7830973

CCOc1nc2ccccc2cc1C#N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.56
GAA P10253 5/20 0.56
KDM4E B2RXH2 7/20 0.53
L3MBTL1 Q9Y468 1/20 0.50
TLR8 Q9NR97 2/20 0.49
MAPT P10636 7/20 0.46
HPGD P15428 4/20 0.46
TSHR P16473 4/20 0.46
TDP1 Q9NUW8 2/20 0.46
TP53 P04637 1/20 0.46
ALOX15 P16050 1/20 0.46
HBB P68871 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CASP1 P29466 4/20 0.45
CASP7 P55210 3/20 0.45
HSD17B10 Q99714 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
LMNA P02545 1/20 0.45
PIP4K2A P48426 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30222305 0.88 TLR8 (0.51) ALDH1A1GAAKDM4EL3MBTL1TLR8
SCHEMBL28751326 0.85 GAA (0.50) ALDH1A1GAAKDM4ETLR8MAPT
SCHEMBL27498521 0.84 TSHR (0.54) ALDH1A1GAAKDM4ETLR8MAPT
SCHEMBL29528942 0.82 KDM4E (0.57) ALDH1A1GAAKDM4EL3MBTL1TLR8
SCHEMBL8000025 0.82 KDM4E (0.57) ALDH1A1GAAKDM4EL3MBTL1TLR8
SCHEMBL18023063 0.77 ALDH1A1 (0.62) ALDH1A1GAAKDM4ETLR8MAPT
SCHEMBL28310888 0.77 TLR8 (0.68) ALDH1A1GAAKDM4EL3MBTL1TLR8
SCHEMBL31167298 0.76 MEN1 (0.49) ALDH1A1GAAKDM4EMAPTHPGD
SCHEMBL18023045 0.76 ALDH1A1 (0.60) ALDH1A1GAAKDM4ETLR8MAPT
SCHEMBL18641090 0.76 ALDH1A1 (0.65) ALDH1A1GAAKDM4ETLR8MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103965120-B Quinoline and quinazoline derivant, preparation method, intermediate, compositions and application 上海医药集团股份有限公司 2016-08-17 CN disclosed
US-6288082-B1 COMPOUNDS SUCH AS 6,7-DIETHOXY-4-(INDAN-5-YLAMINO) -QUINOLINE-3-CARBONITRILE USED AS ANTINEOPLASTIC AGENTS AND IN THE TREATMENT OF POLYCYCSTIC KIDNEY DISEASE AMERICAN CYANAMID COMPANY 2001-09-11 US disclosed
EP-1117659-A1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS American Cyanamid Company (US) 2001-07-25 EP disclosed
WO-2000018761-A1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-04-06 WO disclosed