SCHEMBL7831016

SCHEMBL7831016

O=C(O)CCc1nccc(-c2ccc([N+](=O)[O-])cc2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 1/20 0.47
GABRA1 P14867 1/20 0.46
GABRB2 P47870 1/20 0.46
PIK3CA P42336 4/20 0.45
PIK3CB P42338 4/20 0.45
PIK3CG P48736 4/20 0.45
ALDH1A1 P00352 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
MAPT P10636 3/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
FOLH1 Q04609 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TYMP P19971 1/20 0.40
FBP1 P09467 1/20 0.40
PPARG P37231 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40
PLK1 P53350 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203064 0.78 MAPT (0.54) LTB4RGABRA1GABRB2ALDH1A1MAPT
SCHEMBL5206981 0.77 MAPT (0.51) LTB4RGABRA1GABRB2ALDH1A1SMN1; SMN2
SCHEMBL4530760 0.74 PIK3CA (0.48) PIK3CAPIK3CBPIK3CGALDH1A1SMN1; SMN2
SCHEMBL17983523 0.74 TYMP (0.60) GABRA1GABRB2MAPTRAB9ANPC1
SCHEMBL21373454 0.73 PIK3CA (0.60) PIK3CAPIK3CBPIK3CGALDH1A1MAPT
SCHEMBL2369694 0.71 PIK3CA (0.57) PIK3CAPIK3CBPIK3CGMAPTRAB9A
SCHEMBL4526945 0.71 ROCK1 (0.57) PIK3CAPIK3CBPIK3CGALDH1A1MAPT
SCHEMBL350869 0.70 TSHR (0.63) ALDH1A1SMN1; SMN2MAPTRAB9ANPC1
SCHEMBL28712359 0.69 PIK3CA (0.46) PIK3CAPIK3CBPIK3CGALDH1A1SMN1; SMN2
SCHEMBL6385895 0.69 FBP1 (0.50) GABRA1GABRB2ALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131288-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-09-12 EP disclosed
US-6166015-A Pyrrolidine derivatives-CCR-3 receptor antagonists SYNTEX (U.S.A.) INC. (US) 2000-12-26 US disclosed
WO-2000031032-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-02 WO disclosed