SCHEMBL7831019

SCHEMBL7831019

CCCCCc1[c]ccc([N+](=O)[O-])c1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.43
ESPL1 Q14674 1/20 0.40
MAPT P10636 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP19A1 P11511 4/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL231178 0.89 KDM4E (0.42) ESPL1MAPTALDH1A1TDP1CYP1A2
SCHEMBL458041 0.82 POLB (0.43) MAPTALDH1A1TDP1CYP1A2
SCHEMBL8182516 0.79 KMT2A (0.38) MAPTALDH1A1TDP1CYP1A2
SCHEMBL27773763 0.79 TSHR (0.39) KCNH2ALDH1A1TDP1CYP1A2
SCHEMBL5742336 0.78 HTT (0.38) MAPTALDH1A1TDP1CYP1A2
SCHEMBL11286333 0.78 TSHR (0.45) ALDH1A1TDP1CYP1A2CYP19A1
SCHEMBL9625596 0.77 ALDH1A1 (0.37) KCNH2ALDH1A1TDP1CYP1A2CYP19A1
SCHEMBL6377117 0.75 TSHR (0.49) MAPTALDH1A1TDP1CYP1A2
SCHEMBL7304803 0.75 TSHR (0.42) ALDH1A1TDP1CYP1A2
SCHEMBL5585098 0.75 LOXL2 (0.46) MAPTALDH1A1TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2332940-B1 Azaindoles useful as inhibitors of JAK and other protein kinases VERTEX PHARMA (US) 2012-10-31 EP claimed
EP-0699676-B1 Physical form of dihidro-2,3-benzodiazepine derivative LILLY CO ELI (US) 2001-02-07 EP claimed