SCHEMBL7832308

SCHEMBL7832308

CCOC(=O)c1cn(-c2nccs2)c2nc(N3CC(NCC(=O)OC(C)(C)C)C(OC)C3)ccc2c1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 2/20 0.34
RXFP1 Q9HBX9 1/20 0.33
KDM4E B2RXH2 3/20 0.33
HPGD P15428 2/20 0.33
CYP2C19 P33261 1/20 0.33
CSF1R P07333 1/20 0.33
ALDH1A1 P00352 3/20 0.32
ATM Q13315 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
TYK2 P29597 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
RET P07949 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7832305 1.00 OPRK1 (0.34) OPRK1RXFP1KDM4EHPGDCYP2C19
SCHEMBL7832312 1.00 OPRK1 (0.34) OPRK1RXFP1KDM4EHPGDCYP2C19
SCHEMBL7835604 0.92 HTR3A (0.32) KMT2AMEN1LMNARETHTR3A
SCHEMBL7835607 0.92 HTR3A (0.32) KMT2AMEN1LMNARETHTR3A
SCHEMBL7835615 0.92 HTR3A (0.32) KMT2AMEN1LMNARETHTR3A
SCHEMBL7823053 0.90 OPRK1 (0.32) OPRK1RXFP1KDM4EHPGDCYP2C19
SCHEMBL708977 0.89 RXFP1 (0.37) OPRK1RXFP1KDM4EHPGDCYP2C19
SCHEMBL7831785 0.89 RXFP1 (0.37) OPRK1RXFP1KDM4EHPGDCYP2C19
SCHEMBL7831769 0.89 RXFP1 (0.37) OPRK1RXFP1KDM4EHPGDCYP2C19
SCHEMBL8802441 0.87 RET (0.31) RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0787726-B1 NOVEL COMPOUND, PROCESS FOR PRODUCING THE SAME, AND ANTITUMOR AGENT DAINIPPON PHARMACEUTICAL CO (JP) 2001-11-28 EP disclosed
EP-0787726-A1 NOVEL COMPOUND, PROCESS FOR PRODUCING THE SAME, AND ANTITUMOR AGENT DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1997-08-06 EP disclosed