SCHEMBL7832387

SCHEMBL7832387

COc1ccc2cc(-c3ncccc3CO)ccc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 8/20 0.58
CYP11B1 P15538 7/20 0.58
CYP17A1 P05093 3/20 0.51
CYP19A1 P11511 2/20 0.51
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 2/20 0.50
HPGD P15428 1/20 0.50
RAB9A P51151 3/20 0.48
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
KCNA5 P22460 1/20 0.47
TEK Q02763 1/20 0.46
HSD17B1 P14061 1/20 0.45
HSD17B2 P37059 1/20 0.45
NPC1 O15118 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16048953 0.86 KDM4E (0.66) CYP11B2CYP11B1KDM4EALDH1A1HPGD
SCHEMBL16047508 0.85 KCNA5 (0.62) CYP19A1KDM4EALDH1A1HPGDKCNA5
SCHEMBL11620358 0.79 KDM4E (0.55) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL5749914 0.79 CYP11B2 (0.50) CYP11B2CYP11B1CYP17A1CYP19A1KDM4E
SCHEMBL8318119 0.77 KDM4E (0.49) KDM4EALDH1A1HPGDRAB9AMEN1
SCHEMBL31536244 0.75 CYP11B2 (0.55) CYP11B2CYP11B1CYP17A1CYP19A1KDM4E
SCHEMBL4114679 0.74 SYK (0.56) ALDH1A1RAB9ANPC1
SCHEMBL6338303 0.73 CYP17A1 (0.57) CYP11B2CYP11B1CYP17A1CYP19A1TEK
SCHEMBL17084671 0.73 ALDH1A1 (0.59) CYP11B2CYP11B1KDM4EALDH1A1HPGD
SCHEMBL16046684 0.73 KDM4E (0.59) KDM4EALDH1A1HPGDRAB9AKCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073640-A1 NAPHTHALENE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2001-02-07 EP disclosed
WO-1999054309-A1 NAPHTHALENE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-10-28 WO disclosed