SCHEMBL7832660

SCHEMBL7832660

CNC(=O)c1c(C)[nH]c2ccc(O)c(CN(C)C)c12

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.46
KMT2A Q03164 5/20 0.43
MEN1 O00255 4/20 0.43
TSHR P16473 3/20 0.43
LMNA P02545 2/20 0.43
ALDH1A1 P00352 3/20 0.40
PKM P14618 1/20 0.40
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.39
GRIN2B Q13224 1/20 0.39
EP300 Q09472 2/20 0.39
CREBBP Q92793 2/20 0.39
BRD4 O60885 1/20 0.39
BRPF1 P55201 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
BRD9 Q9H8M2 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7838453 0.88 ADRB2 (0.49) ADRB2KMT2AMEN1TSHRLMNA
SCHEMBL7832726 0.87 ADRB2 (0.44) ADRB2KMT2AMEN1TSHRLMNA
SCHEMBL7832340 0.84 TSHR (0.48) ADRB2KMT2AMEN1TSHRLMNA
SCHEMBL7827109 0.82 MAPT (0.47) ADRB2KMT2AMEN1TSHRLMNA
SCHEMBL7835197 0.81 TSHR (0.46) ADRB2KMT2AMEN1TSHRLMNA
SCHEMBL7832805 0.81 TSHR (0.62) ADRB2KMT2AMEN1TSHRLMNA
SCHEMBL7837273 0.80 TSHR (0.45) ADRB2KMT2AMEN1TSHRLMNA
SCHEMBL7831675 0.79 GAA (0.48) ADRB2KMT2AMEN1TSHRLMNA
SCHEMBL5324128 0.78 BRD4 (0.36) KMT2AMEN1ALDH1A1PKMHTR2A
SCHEMBL7837276 0.78 TSHR (0.50) ADRB2KMT2AMEN1TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144415-A2 FUNCTIONALIZED HETEROCYCLES AS CHEMOKINE RECEPTOR MODULATORS WARNER-LAMBERT COMPANY (US) 2001-10-17 EP disclosed
WO-2000042045-A2 FUNCTIONALIZED HETEROCYCLES AS CHEMOKINE RECEPTOR MODULATORS WARNER-LAMBERT COMPANY (US) 2000-07-20 WO disclosed