SCHEMBL7833808

SCHEMBL7833808

O=C(O)C#Cc1cccc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.47
NR4A2 P43354 1/20 0.47
NR4A3 Q92570 1/20 0.47
CHAT P28329 1/20 0.44
TDP1 Q9NUW8 2/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
ACACB O00763 1/20 0.42
PTPN1 P18031 1/20 0.42
CDC25B P30305 1/20 0.42
GRM5 P41594 1/20 0.41
MAPT P10636 2/20 0.40
HTT P42858 2/20 0.40
WDR5 P61964 1/20 0.40
MEN1 O00255 1/20 0.40
MITF O75030 1/20 0.40
RAD52 P43351 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29749080 1.00 NR4A1 (0.47) NR4A1NR4A2NR4A3CHATTDP1
SCHEMBL30772315 0.81 HSP90AA1 (0.48) TDP1CA1CA2PTPN1MAPT
SCHEMBL6561814 0.79 PLK1 (0.49) NR4A1NR4A2NR4A3CHATCA1
SCHEMBL29661843 0.79 CHAT (0.60) CHATTDP1CA1CA2ACACB
SCHEMBL2776015 0.79 CHAT (0.60) CHATTDP1CA1CA2ACACB
SCHEMBL3130959 0.78 NR4A1 (0.63) NR4A1NR4A2NR4A3CHATTDP1
SCHEMBL5881377 0.77 CA1 (0.50) NR4A1NR4A2NR4A3CHATTDP1
SCHEMBL6364668 0.77 CHAT (0.58) CHATTDP1CA1CA2ACACB
SCHEMBL5881381 0.75 CHAT (0.49) NR4A1NR4A2NR4A3CHATTDP1
SCHEMBL5881479 0.75 CHAT (0.49) CHATTDP1CA1CA2ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113548965-B Preparation method of 1,4 eneyne compound 南京工业大学 2022-07-26 CN claimed
CN-113429285-B Method for synthesizing hydroxyacetone ester compounds based on methylene aziridine 潍坊科技学院 2021-12-07 CN claimed
CN-113548965-A Preparation method of 1, 4-eneyne compound 南京工业大学 2021-10-26 CN claimed
CN-113429285-A Method for synthesizing hydroxyacetone ester compounds based on methylene aziridine 潍坊科技学院 2021-09-24 CN claimed
CN-115286555-A Synthetic method of 3-alkynylselendole compound 温州医科大学 2022-11-04 CN disclosed
CN-113548965-B Preparation method of 1,4 eneyne compound 南京工业大学 2022-07-26 CN disclosed
CN-113349200-B Application of magnolol and honokiol as pesticide synergist 中国水稻研究所 2022-05-24 CN disclosed
CN-113429285-B Method for synthesizing hydroxyacetone ester compounds based on methylene aziridine 潍坊科技学院 2021-12-07 CN disclosed
CN-113548965-A Preparation method of 1, 4-eneyne compound 南京工业大学 2021-10-26 CN disclosed
CN-113429285-A Method for synthesizing hydroxyacetone ester compounds based on methylene aziridine 潍坊科技学院 2021-09-24 CN disclosed
CN-113349200-A Application of magnolol and honokiol as pesticide synergist 中国水稻研究所 2021-09-07 CN disclosed
US-6300340-B1 USEFUL FOR THERAPY OF CANCER AND SOLID TUMORS ADIR ET COMPAGNIE (FR) 2001-10-09 US disclosed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
US-6162822-A Bisimide compounds ADIR ET COMPAGNIE (FR) 2000-12-19 US disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed
US-5854273-A Bisimide compounds ADIR ET COMPAGNIE (FR) 1998-12-29 US disclosed