SCHEMBL7833982

SCHEMBL7833982

Nc1nc(Cc2ccc3c(c2)=CC(=O)N=3)nc2nc[nH]c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.39
GDA Q9Y2T3 1/20 0.39
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
POLA1 P09884 2/20 0.36
PIN1 Q13526 5/20 0.34
PNP P00491 1/20 0.34
CDK2 P24941 4/20 0.33
MGMT P16455 3/20 0.33
CDK1 P06493 3/20 0.33
CCNB1 P14635 3/20 0.33
CCNA2 P20248 3/20 0.33
CCNA1 P78396 3/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7822337 0.99 PDPK1 (0.38) PDPK1GDAPDE4APDE4BPDE4C
SCHEMBL29557469 0.73 PDE4A (0.64) PDPK1GDAPDE4APDE4BPDE4C
SCHEMBL104931 0.73 PDE4A (0.64) PDPK1GDAPDE4APDE4BPDE4C
SCHEMBL7822681 0.72 NEK2 (0.46) PDPK1GDAPDE4APDE4BPDE4C
SCHEMBL7833385 0.72 MPO (0.45) PDPK1GDAPDE4APDE4BPDE4C
SCHEMBL448639 0.72 CDC7 (0.47) PDPK1GDAPDE4APDE4BPDE4C
SCHEMBL288236 0.72 BRAF (0.48) PDPK1GDAPDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL7834487 0.71 MPO (0.44) PDPK1GDAPDE4APDE4BPDE4C
SCHEMBL7840697 0.70 CDC7 (0.57) PDPK1PIN1CDK2MGMTCDK1
SCHEMBL1980128 0.70 PDPK1 (0.45) PDPK1GDAPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP disclosed