SCHEMBL7834583

SCHEMBL7834583

CN(C)c1ncc(-c2cccc(Nc3ccc(-c4ccoc4)cc3N)c2)cn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
CYP2D6 P10635 4/20 0.37
CYP2C19 P33261 4/20 0.37
CYP1A2 P05177 3/20 0.37
CYP3A4 P08684 3/20 0.37
CLK4 Q9HAZ1 3/20 0.37
LMNA P02545 2/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
USP2 O75604 3/20 0.37
TSHR P16473 1/20 0.37
HDAC1 Q13547 1/20 0.36
CNR1 P21554 1/20 0.36
SERPINE1 P05121 1/20 0.36
DHFR P00374 1/20 0.36
FYN P06241 2/20 0.36
HDAC2 Q92769 3/20 0.35
MAP4K4 O95819 3/20 0.35
TGFBR1 P36897 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2643742 0.90 MAP4K4 (0.42) ALDH1A1CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL2643726 0.84 ALK (0.42) DHFRHDAC2HDAC3ALK
SCHEMBL7834274 0.84 AKR1B1 (0.36) ALDH1A1CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL8323635 0.80 DHFR (0.40) DHFRMAP4K4
SCHEMBL9071943 0.79 HDAC2 (0.41) ALDH1A1CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL2643656 0.77 HDAC2 (0.41) ALDH1A1CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL2643659 0.77 HDAC2 (0.43) ALDH1A1CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL7820330 0.74 MAPT (0.40) ALDH1A1CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL2643607 0.74 HDAC2 (0.39) ALDH1A1CYP2D6CYP2C19CYP1A2CYP3A4
SCHEMBL2643125 0.73 SYK (0.37) ALDH1A1CYP2D6CYP2C19CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1164134-A1 Benzimidazole compounds and their use as modulators of the GABA A receptor complex NEUROSEARCH A/S (DK) 2001-12-19 EP disclosed
EP-0821684-B1 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS MODULATORS OF THE GABA A? RECEPTOR COMPLEX NEUROSEARCH AS (DK) 2001-12-05 EP disclosed
US-5922724-A Benzimidazole compounds and their use as modulators of the GABA a receptor complex NEUROSEARCH A/S (DK) 1999-07-13 US disclosed