SCHEMBL8323635

SCHEMBL8323635

CN(C)c1ncc(-c2cccc(Nc3ccc(-n4cccc4)cc3N)c2)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.40
MAP4K4 O95819 2/20 0.33
EGFR P00533 2/20 0.32
GAA P10253 2/20 0.31
MAPT P10636 1/20 0.31
KDM4E B2RXH2 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
NPC1 O15118 1/20 0.31
GFER P55789 1/20 0.31
CDK1 P06493 1/20 0.31
CDK4 P11802 1/20 0.31
CDK2 P24941 1/20 0.31
SYK P43405 1/20 0.31
PRMT5 O14744 1/20 0.30
WDR77 Q9BQA1 1/20 0.30
TYK2 P29597 1/20 0.30
PDE4D Q08499 1/20 0.30
SIRT2 Q8IXJ6 1/20 0.30
SIRT1 Q96EB6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2647222 0.83 CNR1 (0.38) DHFREGFRGAAMAPTKDM4E
SCHEMBL5755261 0.83 L3MBTL1 (0.39) MAPTL3MBTL1
SCHEMBL7834583 0.80 ALDH1A1 (0.37) DHFRMAP4K4
SCHEMBL2647045 0.80 MEN1 (0.43) DHFREGFRABL1PDGFRBBCR
SCHEMBL2643726 0.77 ALK (0.42) DHFREGFR
SCHEMBL2647429 0.76 RET (0.42) DHFRGAANPSR1NPC1CDK1
SCHEMBL2655356 0.70 ABL1 (0.47) MAPTSYKABL1PDGFRBBCR
SCHEMBL2643742 0.69 MAP4K4 (0.42) MAP4K4GAAMAPTKDM4EL3MBTL1
SCHEMBL2643607 0.69 HDAC2 (0.39) GAAMAPTKDM4EL3MBTL1NPC1
SCHEMBL2643560 0.67 MAP4K4 (0.65) DHFRMAP4K4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5902813-A MODULATORS OF THE BENZODIAXEPINE RECEPTOR OT THE GAMMA-BUTYRIC ACID(A) RECEPTOR COMPLEX; ANXIOLYTIC, ANTIEPILEPTIC AND -CONVULSANT AGENTS; SLEEP AND MEMORY DISORDERS NEUROSEARCH A/S (DK) 1999-05-11 US disclosed