SCHEMBL78348

SCHEMBL78348

CC(C(=O)N1CN(C(=O)C(C)c2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)CN(C(=O)C(C)c2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)C1)c1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1A O00555 1/20 0.41
CACNA2D1 P54289 1/20 0.41
CACNB1 Q02641 1/20 0.41
CA2 P00918 2/20 0.41
CA1 P00915 1/20 0.41
LMNA P02545 2/20 0.41
RECQL P46063 1/20 0.41
ALDH1A1 P00352 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
GAA P10253 2/20 0.40
POLB P06746 1/20 0.40
TYR P14679 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
GLRA3 O75311 1/20 0.40
GLRB P48167 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
ALOX5 P09917 1/20 0.39
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7185804 0.90 CACNA1A (0.37) CACNA1ACACNA2D1CACNB1CA2CA1
SCHEMBL6360901 0.85 CACNA1A (0.39) CACNA1ACACNA2D1CACNB1CA2CA1
SCHEMBL8606475 0.84 GAA (0.44) CACNA1ACACNA2D1CACNB1CA2CA1
SCHEMBL11702172 0.79 CA2 (0.50) CA2CA1LMNARECQLALDH1A1
SCHEMBL8466395 0.79 CYP3A4 (0.45) CA2CA1LMNARECQLALDH1A1
SCHEMBL7191036 0.78 CACNA1A (0.33) CACNA1ACACNA2D1CACNB1LMNAALDH1A1
SCHEMBL7196940 0.78 MEN1 (0.33) CACNA1ACACNA2D1CACNB1LMNARECQL
SCHEMBL100584 0.78 GLRA3 (0.50) CACNA1ACACNA2D1CACNB1CA2CA1
SCHEMBL6275312 0.78 GLRA3 (0.50) CACNA1ACACNA2D1CACNB1CA2CA1
SCHEMBL9340528 0.78 CA2 (0.48) CA2CA1LMNARECQLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2177 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240294732-A1 COMPOSITIONS AND METHODS FOR PROTECTING ORGANIC POLYMERIC MATERIALS FROM DISCOLORATION DUE TO EXPOSURE TO UV-C LIGHT CYTEC INDUSTRIES INC. (US) 2024-09-05 US claimed
US-20240182674-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, STABILIZER COMPOSITION, MASTER BATCH OR CONCENTRATE, STABILIZED PLASTIC COMPOSITION, PROCESS FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, AND USE OF COMPOSITIONS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-06-06 US claimed
US-20240174839-A1 STABILIZER MIXTURE BASF SE (DE) 2024-05-30 US claimed
EP-4308638-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING POLYOLEFIN RECYCLATES, STABILIZER COMPOSITION, MASTER BATCH CONCENTRATE, PLASTIC COMPOSITION, MOLDING COMPOUND OR MOLDING, METHOD FOR STABILIZING A POLYOLEFIN RECYCLATE AND USE OF A PLASTIC COMPOSITION Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-24 EP claimed
EP-4301809-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, STABILIZER COMPOSITION, MASTER BATCH OR CONCENTRATE, STABILIZED PLASTIC COMPOSITION, PROCESS FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, AND USE OF COMPOSITIONS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-10 EP claimed
EP-4251689-A1 COMPOSITIONS AND METHODS FOR PROTECTING ORGANIC POLYMERIC MATERIALS FROM DISCOLORATION DUE TO EXPOSURE TO UV-C LIGHT Cytec Industries, Inc. (US) 2023-10-04 EP claimed
WO-2022194672-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING POLYOLEFIN RECYCLATES, STABILIZER COMPOSITION, MASTER BATCH CONCENTRATE, PLASTIC COMPOSITION, MOLDING COMPOUND OR MOLDING, METHOD FOR STABILIZING A POLYOLEFIN RECYCLATE AND USE OF A PLASTIC COMPOSITION Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2022-09-22 WO claimed
WO-2022115573-A1 COMPOSITIONS AND METHODS FOR PROTECTING ORGANIC POLYMERIC MATERIALS FROM DISCOLORATION DUE TO EXPOSURE TO UV-C LIGHT CYTEC INDUSTRIES INC. (US) 2022-06-02 WO claimed
US-9181481-B2 Liquid crystal display device and method of manufacturing the same SAMSUNG DISPLAY CO., LTD. (KR) 2015-11-10 US claimed
EP-1925628-A1 Process for polyolefin silane crosslinking Ciba Holding Inc. (CH) 2008-05-28 EP claimed
EP-0905180-B1 Dust free stabiliser granules containing epoxide and process of their preparation CIBA SC HOLDING AG (CH) 2003-05-21 EP claimed
US-20010044518-A1 Plastic additives, comprising a phenolic antioxidant, organic phosphite or phosphonite, a phosphonate, a sterically hindered amine or a UV absorber, or mixture thereof, and an epoxy compound solid at room temperature HOFFMANN KURT (DE) 2001-11-22 US claimed
EP-0775719-A2 Process for preparing vulcanizable elastomeric compounds from granular elastomer blends UNION CARBIDE CHEMICALS & PLASTICS TECHNOLOGY CORPORATION (US) 1997-05-28 EP claimed
EP-4359495-B1 O-ALKYLATED STERICALLY HINDERED ANTIOXIDANTS SONGWON IND CO LTD (KR) 2026-05-06 EP disclosed
EP-4722284-A1 LOW MELTING CARBOXAMIDE HALS FOR IMPROVED STABILIZATION OF POLYMERS OR RESINS CLARIANT INTERNATIONAL LTD (CH) 2026-04-08 EP disclosed
EP-4722276-A1 LOW MELTING CARBOXAMIDE HALS FOR IMPROVED STABILIZATION OF POLYAMIDES CLARIANT INTERNATIONAL LTD (CH) 2026-04-08 EP disclosed
US-4006140-A AGING RESISTANCE IMPROVERS FOR VULCANIZABLE RUBBERS THE B. F. GOODRICH COMPANY (US) 1977-02-01 US disclosed
US-3978156-A POLY-HYDRAZIDE, PHENOLIC STABILIZER THE B. F. GOODRICH COMPANY (US) 1976-08-31 US disclosed
US-3965077-A VULCANIZATION RETARDERS THE B. F. GOODRICH COMPANY (US) 1976-06-22 US disclosed
US-3957721-A Stabilizer combinations of (β-aminoacrlyl compounds and phenolic compounds and stabilized compositions thereof THE B. F. GOODRICH COMPANY (US) 1976-05-18 US disclosed