SCHEMBL7834898

SCHEMBL7834898

CN(C)c1ccc2c(c1)c(C=O)cn2C

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.62
KDM4E B2RXH2 5/20 0.62
IMPDH2 P12268 1/20 0.56
CYP2A6 P11509 1/20 0.39
CYP2A13 Q16696 1/20 0.39
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
LMNA P02545 1/20 0.37
GAA P10253 2/20 0.36
GLA P06280 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
BCHE P06276 2/20 0.36
IP6K1 Q92551 1/20 0.36
MEN1 O00255 3/20 0.35
POLB P06746 3/20 0.35
RAB9A P51151 3/20 0.35
KMT2A Q03164 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7832439 0.87 ALDH1A1 (0.59) ALDH1A1KDM4EIMPDH2CYP2A6CYP2A13
SCHEMBL30995729 0.80 ALDH1A1 (0.70) ALDH1A1KDM4EIMPDH2HSD17B10MAPT
SCHEMBL2275437 0.80 ALDH1A1 (0.70) ALDH1A1KDM4EIMPDH2HSD17B10MAPT
SCHEMBL1092202 0.77 ALDH1A1 (1.00) ALDH1A1KDM4EIMPDH2LMNASMN1; SMN2
SCHEMBL13363658 0.77 ALDH1A1 (0.66) ALDH1A1KDM4EIMPDH2HPGDHSD17B10
SCHEMBL1450678 0.77 ALDH1A1 (0.66) ALDH1A1KDM4EIMPDH2BCHE
SCHEMBL5437254 0.77 ALDH1A1 (0.66) ALDH1A1KDM4EIMPDH2CYP2A6GSK3B
SCHEMBL1093666 0.77 ALDH1A1 (0.66) ALDH1A1KDM4EIMPDH2MEN1POLB
SCHEMBL1093582 0.74 ALDH1A1 (0.77) ALDH1A1KDM4EIMPDH2BCHEMEN1
SCHEMBL16619395 0.73 ALDH1A1 (0.65) ALDH1A1KDM4EIMPDH2LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680950-B1 PROPENONE DERIVATIVES KYOWA HAKKO KOGYO KK (JP) 2001-05-23 EP disclosed
US-5952355-A 1-ETHER-SUBSTITUTED PHENYL-3-INDOL-3-YL-2-PROPEN-1-ONE DERIVATIVES; ANTITUMOR AND -CARCINOGENIC AGENTS; IMMUNOSUPPRESSANTS; AUTOIMMUNE DISEASES; SIDE EFFECT REDUCTION KYOWA HAKKO KOGYO CO., LTD. (JP) 1999-09-14 US disclosed
EP-0680950-A1 PROPENONE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-11-08 EP disclosed